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183320-51-6

" in MedChemExpress (MCE) Product Catalog:

3

Inhibitors & Agonists

2

Click Chemistry

Art. -Nr. Produktname Target Forschungsgebiete Chemical Structure
  • HY-13256
    Desmethyl Erlotinib hydrochloride
    3 Publications Verification

    OSI-420; CP-373420 hydrochloride

    Drug Metabolite Cancer
    Desmethyl Erlotinib hydrochloride (OSI-420) is an active metabolite of Erlotinib. Erlotinib is a potent EGFR tyrosin kinase inhibitor . Desmethyl Erlotinib (hydrochloride) is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
    Desmethyl Erlotinib hydrochloride
  • HY-13256R

    OSI-420 (Standard); CP-373420 hydrochloride (Standard)

    Reference Standards Drug Metabolite Cancer
    Metoclopramide (hydrochloride hydrate) (Standard) is the analytical standard of Metoclopramide (hydrochloride hydrate). This product is intended for research and analytical applications. Metoclopramide hydrochloride hydrate is a potent antagonist of 5-HT3 and dopamine D2 receptor, with IC50s of 308 nM and 483 nM, respectively. Metoclopramide hydrochloride hydrate can be used for the research of nausea and vomiting, gastro-oesophageal reflux, and gastroparesis .
    Desmethyl Erlotinib hydrochloride (Standard)
  • HY-13256A
    Desmethyl Erlotinib
    3 Publications Verification

    OSI-420 free base; CP-373420

    Drug Metabolite Cancer
    Desmethyl Erlotinib (OSI-420 free base) is an active metabolite of Erlotinib. Erlotinib is a potent EGFR tyrosin kinase inhibitor . Desmethyl Erlotinib is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
    Desmethyl Erlotinib

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