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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
19 Results for "
Antihistamine-1
" in MedChemExpress (MCE) Product Catalog:
Products (19)
19 Results for "Antihistamine-1" in MCE Product Catalog:
Research Areas:
Antihistamine-1 is a H1-antihistamine (Ki=6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel with IC50s of 5.4 and 0.8 μM, respectively.
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Dimenhydrinate is an orally active H1-antihistamine consisting of Diphenhydramine (HY-B0303) and 8-Chlorotheophylline. Dimenhydrinate is used to prevent nausea, vomiting, dizziness, and vertigo associated with motion sickness [1].
Cat. No.: HY-32329A
CAS No.: 85650-57-3
Synonyms: MO-8282
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Setiptiline maleate (MO-8282 maleate) is a serotonin receptor antagonist. Setiptiline maleate is a tetracyclic antidepressant (TeCA) which acts as a noradrenergic and specific serotonergic antidepressant (NaSSA). Setiptiline maleate acts as a norepinephrine reuptake inhibitor, α2-adrenergic receptor antagonist, and serotonin receptor antagonist, likely at the 5-HT2A, 5-HT2C, and/or 5-HT3 subtypes, as well as an H1 receptor inverse agonist/antihistamine .
Cat. No.: HY-100238R
CAS No.: 1186430-60-3
Research Areas:
Antihistamine-1 (Standard) is the analytical standard of Antihistamine-1 (HY-100238). This product is intended for research and analytical applications. Antihistamine-1 is a H1-antihistamine (Ki=6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel with IC50s of 5.4 and 0.8 μM, respectively.
Cat. No.: HY-B0539S3
CAS No.: 1020719-34-9
Synonyms: Sch34117-d5
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Phenindamine (Nu 1504) is an antihistamine .
Cat. No.: HY-B0157AS
CAS No.: 1795138-23-6
Synonyms: HC 20-511-d3 fumarate
Research Areas:
Ketotifen-d3 (fumarate) is the deuterium labeled Ketotifen fumarate. Ketotifen (HC 20511) fumarate is a second-generation noncompetitive H1-antihistamine and mast cell stabilizer, which is used to prevent asthma attacks [1] .
Research Areas:
Dimenhydrinate (Standard) is the analytical standard of Dimenhydrinate. This product is intended for research and analytical applications. Dimenhydrinate is an orally active H1-antihistamine consisting of Diphenhydramine (HY-B0303) and 8-Chlorotheophylline. Dimenhydrinate is used to prevent nausea, vomiting, dizziness, and vertigo associated with motion sickness [1].
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Phenindamine tartrate is a Histamine H1-receptor antagonist. Phenindamine tartrate is an antihistamine .
Cat. No.: HY-W683872
CAS No.: 16188-61-7
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Talastine is a potent H1-antihistamine. Talastine can induce allergic exanthema [1] .
Cat. No.: HY-W281862
CAS No.: 57734-69-7
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Sequifenadine is a H1-antihistamine. Sequifenadine has the potential for the research of inflammatory eye disease with allergic symptoms [1] .
Cat. No.: HY-118910
CAS No.: 119810-68-3
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AHR-14310C is a potent, long-acting, nonsedating H1-antihistamine that prevents antigen-induced mucus formation in sensitive rats [1].
Cat. No.: HY-B0539S1
CAS No.: 1795024-82-6
Synonyms: Sch34117-d9
Cat. No.: HY-B0539S
CAS No.: 381727-29-3
Synonyms: Sch34117-d4
Cat. No.: HY-B0539R
CAS No.: 100643-71-8
Synonyms: Sch34117 (Standard)
Cat. No.: HY-B0539S4
Synonyms: Sch34117-d4 hydrobromide
Cat. No.: HY-B0539S2
CAS No.: 2713301-38-1
Cat. No.: HY-32329S
CAS No.: 1795024-97-3
Cat. No.: HY-32329AR
CAS No.: 85650-57-3
Synonyms: MO-8282 (Standard)
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Research Areas:
Setiptiline (maleate) (Standard) is the analytical standard of Setiptiline (maleate). This product is intended for research and analytical applications. Setiptiline maleate (MO-8282 maleate) is a serotonin receptor antagonist. Setiptiline maleate is a tetracyclic antidepressant (TeCA) which acts as a noradrenergic and specific serotonergic antidepressant (NaSSA). Setiptiline maleate acts as a norepinephrine reuptake inhibitor, α2-adrenergic receptor antagonist, and serotonin receptor antagonist, likely at the 5-HT2A, 5-HT2C, and/or 5-HT3 subtypes, as well as an H1 receptor inverse agonist/antihistamine .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
