6 Results for "

CRHR1 antagonist

" in MedChemExpress (MCE) Product Catalog:
Products (6)

6 Results for "CRHR1 antagonist" in MCE Product Catalog:

  • Targets Recommended:
8
8 Publications Verification
Cat. No.: HY-103377
CAS No.: 220953-69-5
Purity:  99.87%
Target:  

CRFR

Antalarmin (hydrochloride) is an oral active non-peptide corticotropin-releasing hormone receptor 1 (CRHR1) antagonist with a Ki of 1 nM. Antalarmin hydrochloride suppresses CRH-induced ACTH secretion and blocks CRH and novelty induced anxiety-like behavior in animal models. Antalarmin hydrochloride produces anti-inflammatory effects in arthritis models, and suppresses stress-induced gastric ulceration related to irritable bowel syndrome .
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8
8 Publications Verification
Cat. No.: HY-124475
CAS No.: 157284-96-3
Purity:  99.95%
Target:  

CRFR

Research Areas:  

Neurological Disease

Antalarmin is a selective nonpeptide corticotropin-releasing factor receptor 1 (CRHR1) antagonist with a Ki of 2.7 nM. Antalarmin can pass through the blood–brain barrier .
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1
1 Cited Publications
Cat. No.: HY-12131
CAS No.: 202578-52-7
Purity:  98.73%
Target:  

CRFR

Research Areas:  

Neurological Disease Endocrinology

DMP 696 is a selective corticotropin-releasing hormone receptor 1 (CRHR1) antagonist, used for the treatment of anxiety and depression.
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Cat. No.: HY-139035
CAS No.: 276890-57-4
Target:  

CRFR

Research Areas:  

Neurological Disease

CRHR1 antagonist 1 (compound 10a) is a non-peptide corticotropin-releasing hormone type 1 receptor (CRHR1) antagonist. CRHR1 antagonist 1 can be utilized in mental disorders research .
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Cat. No.: HY-124475R
CAS No.: 157284-96-3
Target:  

CRFR

Research Areas:  

Neurological Disease

Antalarmin (Standard) is the analytical standard of Antalarmin. This product is intended for research and analytical applications. Antalarmin is a selective nonpeptide corticotropin-releasing factor receptor 1 (CRHR1) antagonist with a Ki of 2.7 nM. Antalarmin can pass through the blood–brain barrier .
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Cat. No.: HY-103377R
CAS No.: 220953-69-5
Antalarmin (hydrochloride) (Standard) is the analytical standard of Antalarmin (hydrochloride). This product is intended for research and analytical applications. Antalarmin (hydrochloride) is an oral active non-peptide corticotropin-releasing hormone receptor 1 (CRHR1) antagonist with a Ki of 1 nM. Antalarmin hydrochloride suppresses CRH-induced ACTH secretion and blocks CRH and novelty induced anxiety-like behavior in animal models. Antalarmin hydrochloride produces anti-inflammatory effects in arthritis models, and suppresses stress-induced gastric ulceration related to irritable bowel syndrome .
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