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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
16 Results for "
PAC1 receptor
" in MedChemExpress (MCE) Product Catalog:
Products (16)
16 Results for "PAC1 receptor" in MCE Product Catalog:
5
5 Cited Publications
Cat. No.: HY-P0221
CAS No.: 137061-48-4
Synonyms: Pituitary Adenylate Cyclase Activating Polypeptide 38
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3
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3
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2
2 Cited Publications
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PA-8 is a potent, selective and orally active PACAP type I (PAC1) receptor antagonist. PA-8 inhibits the phosphorylation of CREB induced by PACAP in PAC1-, but not VPAC1- or VPAC2-receptor. PA-8 also inhibits PACAP-induced cAMP elevation with an IC50 of 2 nM .
1
1 Cited Publications
Synonyms: PAC1R antagonist 1
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PA-915 (PAC1R antagonist 1) is a potent and orally active antagonist of PAC1 receptor. PA-915 inhibits pituitary adenylate cyclase-activating polypeptide (PACAP)-induced CREB phosphorylation. PA-915 can inhibit PACAP- and nerve injury-induced allodynia. PA-915 can be used for the research of neuropathic pain .
Cat. No.: HY-P99509
CAS No.: 2225850-33-7
Synonyms: AMG-301
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Cat. No.: HY-P0221C
CAS No.: 129405-61-4
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PA-9 is a pituitary adenylate cyclase-activating polypeptide (PACAP) type I (PAC1) receptor antagonist. PA-9 dose dependently inhibits PACAP-induced cAMP elevation with an IC50 of 5.6 nM. PA-9 can be used for the research of neuropathic and/or inflammatory pain .
Cat. No.: HY-P3483
CAS No.: 135374-80-0
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Cat. No.: HY-P1817
CAS No.: 144025-82-1
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Cat. No.: HY-P0221A
Synonyms: Pituitary Adenylate Cyclase Activating Polypeptide 38 TFA
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Cat. No.: HY-P3483A
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Cat. No.: HY-P1817A
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Cat. No.: HY-P77120A
Purity: ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: ADCYAP1R1; PAC1 receptor; ADCYAP receptor Type I; PACAP-R1; PAC1R; Pituitary Adenylate Cyclase Activating Polypeptide 1 receptor Type I Hiphop Splice Variant; Pituitary Adenylate Cyclase-Activating Polypeptide Type I receptor; Pituitary Adenylate Cyclase
Species:
Human
Source:
HEK293
Cat. No.: HY-P77120
Purity: ≥ 85%, as determined by reducing SDS-PAGE.
Synonyms: ADCYAP1R1; PAC1 receptor; ADCYAP receptor Type I; PACAP-R1; PAC1R; Pituitary Adenylate Cyclase Activating Polypeptide 1 receptor Type I Hiphop Splice Variant; Pituitary Adenylate Cyclase-Activating Polypeptide Type I receptor; Pituitary Adenylate Cyclase
Species:
Human
Source:
HEK293
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
