1436004-46-4
1436004-46-4
Chemical Structure
PA-9
- CAS No.: 1436004-46-4
- Formula:C17H18N6O2
- Molecular Weight:338.36
IUPAC Name: N-(2-(1H-imidazol-5-yl)ethyl)-1-(1H-indazol-3-yl)-5-oxopyrrolidine-3-carboxamide
InChIKey: WWPHFXOMYQJGGF-UHFFFAOYSA-N
SMILES: O=C(C(C1)CN(C2=NNC3=C2C=CC=C3)C1=O)NCCC4=CN=CN4
Biological Activity: PA-9 is a pituitary adenylate cyclase-activating polypeptide (PACAP) type I (PAC1) receptor antagonist. PA-9 dose dependently inhibits PACAP-induced cAMP elevation with an IC50 of 5.6 nM. PA-9 can be used for the research of neuropathic and/or inflammatory pain[1].
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PA-9 | 99.73% | PA-9 is a pituitary adenylate cyclase-activating polypeptide (PACAP) type I (PAC1) receptor antagonist. PA-9 dose dependently inhibits PACAP-induced cAMP elevation with an IC50 of 5.6 nM. PA-9 can be used for the research of neuropathic and/or inflammatory pain. | ||||||||||||||||||||
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References
Keywords
