1. GPCR/G Protein
    Neuronal Signaling
    Immunology/Inflammation
  2. Histamine Receptor
  3. ROS 234 dioxalate

ROS 234 dioxalate 

Cat. No.: HY-107563A
Handling Instructions

ROS 234 dioxalate is a potent H3 antagonist, with a pKB of 9.46 for Guinea-pig ileum H3-receptor, a pKi of 8.90 for Rat cerebral cortex H3-receptor, and a ED50 of 19.12 mg/kg (ip) in ex vivo of Rat cerebral cortex. ROS 234 dioxalate diaplays poor central access.

For research use only. We do not sell to patients.

ROS 234 dioxalate Chemical Structure

ROS 234 dioxalate Chemical Structure

CAS No. : 1781941-93-2

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Description

ROS 234 dioxalate is a potent H3 antagonist, with a pKB of 9.46 for Guinea-pig ileum H3-receptor, a pKi of 8.90 for Rat cerebral cortex H3-receptor, and a ED50 of 19.12 mg/kg (ip) in ex vivo of Rat cerebral cortex. ROS 234 dioxalate diaplays poor central access[1][2].

IC50 & Target

H2 Receptor

8.90 (pKi, Rat cerebral cortex H3-receptor)

In Vivo

ROS 234, centrally injected, significantly shortens pentobarbital narcosis[1].

Molecular Weight

421.36

Formula

C₁₇H₁₉N₅O₈

CAS No.

1781941-93-2

SMILES

O=C(O)C(O)=O.O=C(O)C(O)=O.C1(NCCCC2=CN=CN2)=NC3=CC=CC=C3N1

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
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Keywords:

ROS 234 dioxalateHistamine ReceptorInhibitorinhibitorinhibit

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ROS 234 dioxalate
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