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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
7 Results for "
Penbutolol
" in MedChemExpress (MCE) Product Catalog:
Products (7)
7 Results for "Penbutolol" in MCE Product Catalog:
Synonyms: (R)-Penbutolol; (+)-IsoPenbutolol
Target:
Research Areas:
(+)-Penbutolol is a β-adrenoceptor antagonist, with an IC50 of 0.74 μM . (+)-Penbutolol is an optical isomer of l-penbutolol with Na + channel-blocking action .
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1 Cited Publications
Cat. No.: HY-116790
CAS No.: 38363-40-5
Synonyms: (S)-Penbutolol; (-)-IsoPenbutolol
Target:
Research Areas:
(-)-Penbutolol ((S)-Penbutolol) is a potent β-adrenoceptor and 5-HT receptor antagonist with Ki values of 11.6 nM and 11.9 nM for 5-HT in rat cornu ammonis 1 (CA1) and human CA3 .
Cat. No.: HY-116790B
CAS No.: 36507-48-9
Synonyms: (Rac)-Penbutolol; (±)-IsoPenbutolol
Target:
Research Areas:
(±)-Penbutolol ((Rac)-Penbutolol) is the racemic mixture of Penbutolol. (±)-Penbutolol is an orally active β-adrenergic receptor antagonist. (±)-Penbutolol antagonizes exercise-induced tachycardia, reduces the increase in peak expiratory flow rate (PEFR) caused by exercise, and decreases resting plasma renin activity (PRA). (±)-Penbutolol reaches peak plasma concentration 1 hour after oral administration, with a half-life of 4.5 hours, and is converted into an active metabolite in the body. (±)-Penbutolol can be used in cardiovascular-related disease research .
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Penbutolol sulfate ((-)-Terbuclomine) is a potent β-adrenoceptor and 5-HT receptor antagonist with Ki of 11.6 nM and 11.9 nM for 5-HT in rat cornu ammonis 1 (CA1) and human CA3 .
Cat. No.: HY-116790BS
CAS No.: 1346747-40-7
Synonyms: (Rac)-Penbutolol-d9; (±)-IsoPenbutolol-d9
Cat. No.: HY-116790BSA
CAS No.: 1346605-01-3
Synonyms: (Rac)-Penbutolol-d9 hydrochloride; (±)-IsoPenbutolol-d9 hydrochloride
Cat. No.: HY-B1154R
CAS No.: 38363-32-5
Synonyms: (-)-Terbuclomine (Standard)
Research Areas:
Penbutolol (sulfate) (Standard) is the analytical standard of Penbutolol (sulfate). This product is intended for research and analytical applications. Penbutolol sulfate ((-)-Terbuclomine) is a potent β-adrenoceptor and 5-HT receptor antagonist with Ki of 11.6 nM and 11.9 nM for 5-HT in rat cornu ammonis 1 (CA1) and human CA3 .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
