2 Results for "

pyrrolobenzodiazepine dimer cytotoxin

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "pyrrolobenzodiazepine dimer cytotoxin" in MCE Product Catalog:

Cat. No.: HY-161252
CAS No.: 2093165-00-3
Target:  

ADC Payloads

Research Areas:  

Cancer

PBD-monoamide, a modified PBD (pyrrolobenzodiazepine) dimer, is an ADC Cytotoxin. PBD-monoamide can be used for synthesis of DHES0815A (an HER2 ADC). PBD-monoamide has DNA-binding activity and reduces cell viability .
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Cat. No.: HY-P99881
CAS No.: 2095467-44-8
Synonyms: ABBV 176

Research Areas:  

Cancer

Rolinsatamab talirine (ABBV 176) is a prolactin receptor (PRLR)-targeting antibody-drug conjugate (ADC), compoused of Rolinsatamab (HY-P99238) and SGD-1882 (HY-101127). Rolinsatamab talirine binds to PRLR to deliver a cytotoxin to tumor cells. Rolinsatamab talirine induces DNA damage, and exhibits cytotoxicity against multiple breast tumor models, including triple negative and low PRLR-expressing models. Rolinsatamab talirine demonstrates enhanced anti-tumor activity in several breast cancer models. Rolinsatamab talirine can be used for the research of breast cancer, hepatocellular carcinoma, ovarian cancer, endometrial cancer, prostate cancer, colorectal cancer, adrenocortical carcinoma, and solid tumors .
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