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CBP-IN-1 

Cat. No.: HY-111784 Purity: 99.59% ee.: 99.74%
Handling Instructions

CBP-IN-1 is a potent p300/CBP bromodomain inhibitor.

For research use only. We do not sell to patients.

CBP-IN-1 Chemical Structure

CBP-IN-1 Chemical Structure

CAS No. : 2222941-37-7

Size Price Stock Quantity
Free Sample (0.5-1 mg)   Apply now  
10 mM * 1 mL in DMSO USD 271 In-stock
Estimated Time of Arrival: December 31
5 mg USD 230 In-stock
Estimated Time of Arrival: December 31
10 mg USD 400 In-stock
Estimated Time of Arrival: December 31
50 mg USD 1200 In-stock
Estimated Time of Arrival: December 31
100 mg   Get quote  
200 mg   Get quote  

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Customer Review

Based on 1 publication(s) in Google Scholar

Top Publications Citing Use of Products
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Description

CBP-IN-1 is a potent p300/CBP bromodomain inhibitor[1].

IC50 & Target

p300/CBP[1]

Clinical Trial
Molecular Weight

534.60

Formula

C₃₀H₃₂F₂N₄O₃

CAS No.

2222941-37-7

SMILES

O=C1N(C2=CC=C(F)C(F)=C2)[[email protected]](C3=NC4=CC(C5=C(C)ON=C5C)=CC=C4N3[[email protected]]6CC[[email protected]](OC)CC6)CCC1

Shipping

Room temperature in continental US; may vary elsewhere

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 100 mg/mL (187.06 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 1.8706 mL 9.3528 mL 18.7056 mL
5 mM 0.3741 mL 1.8706 mL 3.7411 mL
10 mM 0.1871 mL 0.9353 mL 1.8706 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: ≥ 5.25 mg/mL (9.82 mM); Clear solution

  • 2.

    Add each solvent one by one:  10% DMSO    90% corn oil

    Solubility: ≥ 5.25 mg/mL (9.82 mM); Clear solution

*All of the co-solvents are provided by MCE.
References

Purity: 99.59% ee.: 99.74%

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  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
CBP-IN-1
Cat. No.:
HY-111784
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