1. Signaling Pathways
  2. GPCR/G Protein
  3. PTHR
  4. PTH1R Isoform
  5. PTH1R Agonist

PTH1R Agonist

PTH1R Agonists (5):

Cat. No. Product Name Effect Purity
  • HY-176945
    PTH1R agonist 3
    Agonist
    PTH1R agonist 3 (Example 47) is a parathyroid hormone 1 receptor (PTH1R) agonist with a pEC50 value of less than 6. PTH1R agonist 3 can be used for the study of bone diseases, such as osteoporosis.
  • HY-176944
    PTH1R agonist 2
    Agonist
    PTH1R agonist 2 (example 3) is a parathyroid hormone 1 receptor (PTH1R) agonist. PTH1R agonist 2 can be used for research of hypoparathyroidism and osteoporosis.
  • HY-176943
    PTH1R agonist 1
    Agonist
    PTH1R agonist 1 (Example 2) is a parathyroid hormone 1 receptor (PTH1R) agonist. PTH1R agonist 1 can be used for research of hypoparathyroidism and osteoporosis.
  • HY-120398
    CH5447240
    Agonist
    CH5447240 is an agonist for parathyroid hormone receptor 1 (PTHR1), that inhibits human PTHR1 with an EC50 of 12 μM. CH5447240 exhibits good metabolic stability in human liver microsomes. CH5447240 increases serum calcium levels in rats. CH5447240 can be used in research about hypoparathyroidism.
  • HY-176946
    PTH1R agonist 4
    Agonist
    PTH1R agonist 4 (Example 63) is a parathyroid hormone 1 receptor (PTH1R) agonist with a pEC50 value greater than 7. PTH1R agonist 4 can be used for the study of bone diseases, such as osteoporosis.