A1/A3 AR antagonist 3
A1/A3 AR antagonist 3 is an A1R/A3R dual antagonist with high affinity at low-micromolar to low-nanomolar. A1/A3 AR antagonist 3 can be used for the research of chronic heart diseases.
For research use only. We do not sell to patients.
- CAS No.: 2665804-57-7
- Formula: C22H19N5O3
- Molecular Weight:401.42
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
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Biological Activity
pKd: 8.25 (A1R); 7.87 (A3R)[1].
pKi: 8.36 (A1R); 8.01 (A3R)[1].
A1/A3 AR antagonist 3 (A17) has binding affinity for A1R and A3R with pKd values of 8.25 and 7.87, respectively[1].
A1/A3 AR antagonist 3 has binding affinity for A1R and A3R with pKi values of 8.36 and 8.01, respectively[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 2665804-57-7
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Molecular Weight 401.42
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Formula C22H19N5O3
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SMILES
N#CC1=CC2=C(NN=C2C3=CC=CC=C3)C(NC4=CC(OC)=C(C(OC)=C4)OC)=N1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
A1/A3 AR antagonist 3 Related Classifications
HY-153333 Related Classifications
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