MAGL-IN-9
MAGL-IN-9 (compound 16) is a selective and reversible MAGL inhibitor with IC50 2.7 nM.
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- CAS No.: 3017151-74-2
- Formule: C25H22F4N2O2S
- Masse moléculaire:490.51
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
- Pureté et documentation
- Références
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Help & FAQs
Activité biologique
Description
IC50 & Target
IC50: 2.7 nM (MAGL)[1]
In Vitro
MAGL-IN-9 (10 μM, 25 min) selectively inhibits MAGL in mouse brain membrane preparations, without affecting other serine hydrolases such as FAAH, ABHD6, and ABHD12[1].
MAGL-IN-9 shows a reversible inhibition mechanism in both preincubation and dilution tests[1].
MAGL-IN-9 inhibits MAGL in U973 cells with an IC50 value of 193 nM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 3017151-74-2
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Masse moléculaire 490.51
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Formule C25H22F4N2O2S
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SMILES
O=C(N1CCC(CC2=CC=C(F)C(SC3=NC=CC(C(F)(F)F)=C3)=C2)CC1)C4=CC=CC(O)=C4
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
MAGL-IN-9 Related Classifications
HY-157040 Related Classifications
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