PF-06655075
Based on 1 Customer Validation
PF-06655075 is a novel andnon–brain-penetrant oxytocin receptor agonist with increased selectivity for the oxytocin receptor and significantly increased pharmacokinetic stability. PF-06655075 can be used as a tool compound to further explore the role of peripheral oxytocin in behavioral response.
Nos produits utilisent uniquement pour la recherche. Nous ne vendons pas aux patients.
- Pureté : 99.65%
- Formule: C75H130N14O22S2
- Masse moléculaire:1644.05
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Stockage:
Sealed storage, away from moisture and light.
Powder -80°C, 2 years , -20°C, 1 year* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)
Activité biologique
Description
IC50 & Target
IC50: OT receptor[1]
Chemical Information
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Appearance Solid
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Masse moléculaire 1644.05
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Formule C75H130N14O22S2
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Color White to off-white
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Sealed storage, away from moisture and light
Powder -80°C 2 years -20°C 1 year * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)
Solvant et solubilité
In Vitro:
DMSO : 100 mg/mL (60.83 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Pureté et documentation
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Fiche technique (277 KB)
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SDS (252 KB)
- English - EN (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Korean - KR (252 KB)
- Portuguese - PT (252 KB)
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Instruction de manipulation (2659 KB)
Références
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 0.6083 mL | 3.0413 mL | 6.0825 mL | 15.2063 mL |
| 5 mM | 0.1217 mL | 0.6083 mL | 1.2165 mL | 3.0413 mL | |
| 10 mM | 0.0608 mL | 0.3041 mL | 0.6083 mL | 1.5206 mL | |
| 15 mM | 0.0406 mL | 0.2028 mL | 0.4055 mL | 1.0138 mL | |
| 20 mM | 0.0304 mL | 0.1521 mL | 0.3041 mL | 0.7603 mL | |
| 25 mM | 0.0243 mL | 0.1217 mL | 0.2433 mL | 0.6083 mL | |
| 30 mM | 0.0203 mL | 0.1014 mL | 0.2028 mL | 0.5069 mL | |
| 40 mM | 0.0152 mL | 0.0760 mL | 0.1521 mL | 0.3802 mL | |
| 50 mM | 0.0122 mL | 0.0608 mL | 0.1217 mL | 0.3041 mL | |
| 60 mM | 0.0101 mL | 0.0507 mL | 0.1014 mL | 0.2534 mL |