1072145-33-5

ERRα antagonist-1 Chemical Structure
1072145-33-5

Chemical Structure

ERRα antagonist-1

  • CAS No.: 1072145-33-5
  • Formula:C21H19N3S2
  • Molecular Weight:377.53

IUPAC Name: (Z)-N-(5H-dibenzo[a,d][7]annulen-5-yl)-3-(4,5-dihydrothiazol-2-yl)thiazolidin-2-imine

InChIKey: OWLQZFQCFCNPKV-LNVKXUELSA-N

SMILES: C12=CC=CC=C1C(/N=C3SCCN\3C4=NCCS4)C5=CC=CC=C5C=C2

Biological Activity: ERRα antagonist-1 (Compound A) is a selective and high affinity agonist for estrogen-related receptor α (ERRα). ERRα antagonist-1 inhibits interaction of ERRα with Proliferator-activated Receptor γ Coactivator-1α (PGC-1α) and PGC-1β, the IC50 values are 170 nM and 180 nM, respectively[1].

Cat. No. Product Name Purity Description Pricing
HY-113960
ERRα antagonist-1 99.57% ERRα antagonist-1 (Compound A) is a selective and high affinity agonist for estrogen-related receptor α (ERRα). ERRα antagonist-1 inhibits interaction of ERRα with Proliferator-activated Receptor γ Coactivator-1α (PGC-1α) and PGC-1β, the IC50 values are 170 nM and 180 nM, respectively.
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This product is a controlled substance and not for sale in your territory.

This product is not for sale in your territory.

This compound is listed in the SVHC (Substances of Very High Concern) candidate list of ECHA (European Chemicals Agency).

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References