1072145-33-5
1072145-33-5
Chemical Structure
ERRα antagonist-1
- CAS No.: 1072145-33-5
- Formula:C21H19N3S2
- Molecular Weight:377.53
IUPAC Name: (Z)-N-(5H-dibenzo[a,d][7]annulen-5-yl)-3-(4,5-dihydrothiazol-2-yl)thiazolidin-2-imine
InChIKey: OWLQZFQCFCNPKV-LNVKXUELSA-N
SMILES: C12=CC=CC=C1C(/N=C3SCCN\3C4=NCCS4)C5=CC=CC=C5C=C2
Biological Activity: ERRα antagonist-1 (Compound A) is a selective and high affinity agonist for estrogen-related receptor α (ERRα). ERRα antagonist-1 inhibits interaction of ERRα with Proliferator-activated Receptor γ Coactivator-1α (PGC-1α) and PGC-1β, the IC50 values are 170 nM and 180 nM, respectively[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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ERRα antagonist-1 | 99.57% | ERRα antagonist-1 (Compound A) is a selective and high affinity agonist for estrogen-related receptor α (ERRα). ERRα antagonist-1 inhibits interaction of ERRα with Proliferator-activated Receptor γ Coactivator-1α (PGC-1α) and PGC-1β, the IC50 values are 170 nM and 180 nM, respectively. | ||||||||||||||||||||
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References
Keywords
