42864-78-8
42864-78-8
Chemical Structure
Bevantolol hydrochloride
- CAS No.: 42864-78-8
- Formula:C20H28ClNO4
- Molecular Weight:381.89
IUPAC Name: 1-((3,4-dimethoxyphenethyl)amino)-3-(m-tolyloxy)propan-2-ol hydrochloride
InChIKey: FJTKCFSPYUMXJB-UHFFFAOYSA-N
SMILES: OC(CNCCC1=CC=C(C(OC)=C1)OC)COC2=CC=CC(C)=C2.[H]Cl
Biological Activity: Bevantolol hydrochloride is a selective β1 and α1-adrenergic receptor antagonist with pKi values of 7.83, 6.9 in rat cerebral cortex, respectively. Bevantolol hydrochloride is a potent Ca2+ antagonist[1][2].
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Bevantolol hydrochloride | 98.98% | Bevantolol hydrochloride is a selective β1 and α1-adrenergic receptor antagonist with pKi values of 7.83, 6.9 in rat cerebral cortex, respectively. Bevantolol hydrochloride is a potent Ca2+ antagonist. | ||||||||||||||||||||
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Bevantolol hydrochloride (Standard) | ≥98% | Bevantolol (hydrochloride) (Standard) is the analytical standard of Bevantolol (hydrochloride). This product is intended for research and analytical applications. Bevantolol hydrochloride is a selective β1 and α1-adrenergic receptor antagonist with pKi values of 7.83, 6.9 in rat cerebral cortex, respectively. Bevantolol hydrochloride is a potent Ca2+ antagonist. | ||||||||||||||||||||
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Bevantolol-d7 hydrochloride | Bevantolol-d7 hydrochloride is the deuterium labeled Bevantolol hydrochloride (HY-121186). Bevantolol hydrochloride is a selective β1 and α1-adrenergic receptor antagonist with pKi values of 7.83, 6.9 in rat cerebral cortex, respectively. Bevantolol hydrochloride is a potent Ca2+ antagonist. | |||||||||||||||||||||
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References
- [1]. M Takita, et al. Selectivity of Bevantolol Hydrochloride Towards Alpha- And Beta-Adrenoceptor Subtypes in Rat Cerebral Cortex. Jpn J Pharmacol. 1992 Feb;58(2):193-6. [Content Brief]
- [2]. Takahiro Horinouchi, et al. Different Changes of Plasma Membrane Beta-Adrenoceptors in Rat Heart After Chronic Administration of Propranolol, Atenolol and Bevantolol. Life Sci. 2007 Jul 12;81(5):399-404. [Content Brief]
