GLP-1 receptor agonist 3
GLP-1 receptor agonist 3 (compound (R)-4A-1) is a GLP-1 receptor agonist (WO2018109607A1), used for diabetes research. compound (S)-4A-1 shows EC50s of 1.1 nM and 13 nM in Clone H6 and Clone C6 cell lines assay, respectively.
For research use only. We do not sell to patients.
- CAS No.: 2230200-09-4
- Formula: C31H30FN5O4
- Molecular Weight:555.60
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
EC50: 1.1 nM (GLP-1 receptor, in Clone H6 cell lines assay) and 13 nM (GLP-1 receptor, in Clone C6 cell lines assay)[1]
Chemical Information
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CAS No. 2230200-09-4
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Molecular Weight 555.60
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Formula C31H30FN5O4
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SMILES
O=C(C1=CC=C2N=C(CN3CCC(C4=NC(OCC5=CC=C(C#N)C=C5F)=CC=C4)CC3)N(C[C@@H]6OCC6)C2=C1)O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)