Glucocorticoid receptor agonist-1 phosphate Gly-Glu-Mal

Cat. No.: HY-400878 Purity: 99.80%: FAQs
Data Sheet SDS COA Handling Instructions

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Glucocorticoid receptor agonist-1 phosphate Gly-Glu-Mal, a glucocorticoid receptor agonist, is a drug-linker conjugate for ADC. Glucocorticoid receptor agonist-1 phosphate Gly-Glu-Mal can be used to synthesize the anti-CD40 antibody agent conjugates (WO2019106608A1; example 9).

For research use only. We do not sell to patients.

Glucocorticoid receptor agonist-1 phosphate Gly-Glu-Mal Chemical Structure

CAS No. : 2345732-83-2

Size	Price	Stock	Quantity
1 mg	USD 615	In-stock	Estimated Time of Arrival: December 31
5 mg	USD 1535	In-stock	Estimated Time of Arrival: December 31
10 mg	USD 2456	In-stock	Estimated Time of Arrival: December 31
50 mg		Get quote
100 mg		Get quote

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Biological Activity
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References
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Description

Molecular Weight

915.87

Formula

C₄₆H₅₀N₃O₁₅P

CAS No.

2345732-83-2

Appearance

Solid

Color

White to off-white

SMILES

O=P(O)(O)OCC([C@]12[C@@]3([C@@]([C@@]4([H])[C@]([C@@]5(C(CC4)=CC(C=C5)=O)C)([H])[C@H](C3)O)([H])C[C@@]1([H])O[C@@H](C6=CC=C(C=C6)CC7=CC(NC([C@H](CCC(O)=O)NC(CN8C(C=CC8=O)=O)=O)=O)=CC=C7)O2)C)=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

4°C, sealed storage, away from moisture and light

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)

Solvent & Solubility

In Vitro:

DMSO : 250 mg/mL (272.96 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions

Concentration Solvent Mass	1 mg	5 mg	10 mg

1 mM	1.0919 mL	5.4593 mL	10.9186 mL
5 mM	0.2184 mL	1.0919 mL	2.1837 mL
10 mM	0.1092 mL	0.5459 mL	1.0919 mL

View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

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Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

This equation is commonly abbreviated as: C₁V₁ = C₂V₂

In Vivo Dissolution Calculator

Please enter the basic information of animal experiments:

Dosage

mg/kg

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Dosing volume
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μL

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Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.

Calculation results:

Working solution concentration: mg/mL

Purity & Documentation

Purity: 99.86%

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Data Sheet (273 KB) SDS (0 KB)

COA (258 KB) HNMR (399 KB) RP-HPLC (258 KB) LCMS (103 KB)

Handling Instructions (2659 KB)

References

[1]. Hobson A D, et al. Anti-cd40 antibody drug conjugates. World Intellectual Property Organization. WO2019106608A1.

Complete Stock Solution Preparation Table

Optional Solvent	Concentration Solvent Mass	1 mg	5 mg	10 mg	25 mg

DMSO	1 mM	1.0919 mL	5.4593 mL	10.9186 mL	27.2965 mL
	5 mM	0.2184 mL	1.0919 mL	2.1837 mL	5.4593 mL
	10 mM	0.1092 mL	0.5459 mL	1.0919 mL	2.7296 mL
	15 mM	0.0728 mL	0.3640 mL	0.7279 mL	1.8198 mL
	20 mM	0.0546 mL	0.2730 mL	0.5459 mL	1.3648 mL
	25 mM	0.0437 mL	0.2184 mL	0.4367 mL	1.0919 mL
	30 mM	0.0364 mL	0.1820 mL	0.3640 mL	0.9099 mL
	40 mM	0.0273 mL	0.1365 mL	0.2730 mL	0.6824 mL
	50 mM	0.0218 mL	0.1092 mL	0.2184 mL	0.5459 mL
	60 mM	0.0182 mL	0.0910 mL	0.1820 mL	0.4549 mL
	80 mM	0.0136 mL	0.0682 mL	0.1365 mL	0.3412 mL
	100 mM	0.0109 mL	0.0546 mL	0.1092 mL	0.2730 mL