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Cat. No.: HY-P5897

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GnRH antagonist 3

GnRH antagonist 3 (Compound 11) is a GnRH antagonist with an IC₅₀ of 7 nM. GnRH antagonist 3 can be used in the research of hormone-dependent diseases.

For research use only. We do not sell to patients.

CAS No.: 292141-31-2
Formula: C₄₈H₅₉ClN₁₂O₈
Molecular Weight:967.51

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

GnRH antagonist 3 Chemical Structure

CAS No.: 292141-31-2

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Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- IC₅₀ & Target
Chemical Information
Purity & Documentation
References
Calculators
Help & FAQs
Classifications
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Biological Activity

Description

GnRH antagonist 3 (Compound 11) is a GnRH antagonist with an IC₅₀ of 7 nM. GnRH antagonist 3 can be used in the research of hormone-dependent diseases^[1].

IC₅₀ & Target

IC₅₀: 7 nM (GnRH)^[1]

Chemical Information

CAS No. 292141-31-2
Molecular Weight 967.51
Formula C₄₈H₅₉ClN₁₂O₈
Sequence

Ac-{d-2Nal}-{d-Cpa}-{d-2Pal}-Gly-Arg-Pro-{d-Ala}-NH2
Sequence Shortening

Ac-{d-2Nal}-{d-Cpa}-{d-2Pal}GRPa-NH2
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (258 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Yahalom D, et al. Design and synthesis of potent hexapeptide and heptapeptide gonadotropin-releasing hormone antagonists by truncation of a decapeptide analogue sequence. J Med Chem. 2000 Jul 27;43(15):2831-6. [Content Brief]

Calculators

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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