MGL-IN-2
MGL-IN-2 (Compound 1) is a MGL inhibitor with IC50 values of 0.006 μM and 0.0121 μM for mutant MGL and wild-type MGL, respectively. MGL-IN-2 can be used in the research of metabolic diseases.
For research use only. We do not sell to patients.
- CAS No.: 1252773-92-4
- Formula: C21H18ClF3N4O2S2
- Molecular Weight:514.97
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Description
IC50 & Target
IC50: 0.006 μM and 0.0121 μM for mutant MGL and wild-type MGL, respectively[1]
Chemical Information
-
CAS No. 1252773-92-4
-
Molecular Weight 514.97
-
Formula C21H18ClF3N4O2S2
-
SMILES
O=C(C1=CSC=N1)N2CCN(C3CN(C(C4=C(Cl)C5=CC=C(C(F)(F)F)C=C5S4)=O)C3)CC2
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Protocols
-
Cell Cytotoxicity Assay
Cytotoxicity assays are usually based on the assessment of cell membrane damage, which can also be indirectly detected by measuring cell viability. Detection methods include MTT assay, CKK-8 assay, LDH assay and ATP assay, etc.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)