355367-87-2
Chemical Structure
MEK1 Derived Peptide Inhibitor 1
- CAS 番号: 355367-87-2
- Formula:C68H118N18O17S
- Molecular Weight:1491.84
IUPAC Name: 10-(4-chlorophenyl)-5,5-difluoro-1,3,7,9-tetramethyl-5H-4l4,5l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinine-2-carbaldehyde
InChIKey: AMHJZDPMMQVKID-SOIXIBIBSA-N
SMILES: O=C(N1[C@@H](CCC1)C(N[C@@H](CCCCN)C(N[C@@H](CCCCN)C(N[C@@H](CCCCN)C(N2[C@@H](CCC2)C(N[C@@H]([C@H](O)C)C(N3[C@@H](CCC3)C(N[C@@H]([C@@H](C)CC)C(N[C@@H](CCC(N)=O)C(N[C@@H](CC(C)C)C(N[C@@H](CC(N)=O)C(N4[C@@H](CCC4)C(O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)[C@H](CCSC)N
Biological Activity: MEK1 Derived Peptide Inhibitor 1 is a ERK2 inhibitor that inhibits the activation of ERK2 by MEK1 in vitro, with an IC50 of 30 μM, and exhibits selectivity for ERK over JNK and p38 kinases. MEK1 Derived Peptide Inhibitor 1 can be used to study ERK activation and ERK-mediated responses[1].
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MEK1 Derived Peptide Inhibitor 1 | MEK1 Derived Peptide Inhibitor 1 is a ERK2 inhibitor that inhibits the activation of ERK2 by MEK1 in vitro, with an IC50 of 30 μM, and exhibits selectivity for ERK over JNK and p38 kinases. MEK1 Derived Peptide Inhibitor 1 can be used to study ERK activation and ERK-mediated responses. | |||||||||||||||||||||
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