MAGL-IN-9
MAGL-IN-9 (compound 16) is a selective and reversible MAGL inhibitor with IC50 2.7 nM.
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- CAS 番号: 3017151-74-2
- 分子式: C25H22F4N2O2S
- 分子量:490.51
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
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生物活性
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化学情報
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
生物活性
製品説明
IC50 & Target
IC50: 2.7 nM (MAGL)[1]
体外実験
MAGL-IN-9 (10 μM, 25 min) selectively inhibits MAGL in mouse brain membrane preparations, without affecting other serine hydrolases such as FAAH, ABHD6, and ABHD12[1].
MAGL-IN-9 shows a reversible inhibition mechanism in both preincubation and dilution tests[1].
MAGL-IN-9 inhibits MAGL in U973 cells with an IC50 value of 193 nM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
化学情報
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CAS 番号 3017151-74-2
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分子量 490.51
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分子式 C25H22F4N2O2S
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SMILES
O=C(N1CCC(CC2=CC=C(F)C(SC3=NC=CC(C(F)(F)F)=C3)=C2)CC1)C4=CC=CC(O)=C4
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
MAGL-IN-9 関連分類
HY-157040 関連分類
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