PF-06655075
Based on 1 Customer Validation
PF-06655075 is a novel andnon–brain-penetrant oxytocin receptor agonist with increased selectivity for the oxytocin receptor and significantly increased pharmacokinetic stability. PF-06655075 can be used as a tool compound to further explore the role of peripheral oxytocin in behavioral response.
연구목적의 판매만을 진행합니다. 환자를 대상으로 한 판매는 하지 않습니다.
- Purity : 99.65%
- 화학식: C75H130N14O22S2
- 분자량:1644.05
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보관:
Sealed storage, away from moisture and light.
Powder -80°C, 2 years , -20°C, 1 year* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)
Biological Activity
제품 설명
IC50 & Target
IC50: OT receptor[1]
Chemical Information
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Appearance Solid
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분자량 1644.05
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화학식 C75H130N14O22S2
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Color White to off-white
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선적
Room temperature in continental US; may vary elsewhere.
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보관
Sealed storage, away from moisture and light
Powder -80°C 2 years -20°C 1 year * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)
용액&용해도
In Vitro:
DMSO : 100 mg/mL (60.83 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
순도&문서
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Data Sheet (277 KB)
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SDS (252 KB)
- English - EN (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Korean - KR (252 KB)
- Portuguese - PT (252 KB)
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Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 0.6083 mL | 3.0413 mL | 6.0825 mL | 15.2063 mL |
| 5 mM | 0.1217 mL | 0.6083 mL | 1.2165 mL | 3.0413 mL | |
| 10 mM | 0.0608 mL | 0.3041 mL | 0.6083 mL | 1.5206 mL | |
| 15 mM | 0.0406 mL | 0.2028 mL | 0.4055 mL | 1.0138 mL | |
| 20 mM | 0.0304 mL | 0.1521 mL | 0.3041 mL | 0.7603 mL | |
| 25 mM | 0.0243 mL | 0.1217 mL | 0.2433 mL | 0.6083 mL | |
| 30 mM | 0.0203 mL | 0.1014 mL | 0.2028 mL | 0.5069 mL | |
| 40 mM | 0.0152 mL | 0.0760 mL | 0.1521 mL | 0.3802 mL | |
| 50 mM | 0.0122 mL | 0.0608 mL | 0.1217 mL | 0.3041 mL | |
| 60 mM | 0.0101 mL | 0.0507 mL | 0.1014 mL | 0.2534 mL |