1. Epigenetics
  2. Histone Demethylase
  3. LSD1-IN-7 Methylbenzenesulfonate

LSD1-IN-7 Methylbenzenesulfonate 

Cat. No.: HY-129388
Handling Instructions

LSD1-IN-7 Methylbenzenesulfonate is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity extracted from patent WO2017079670A1, compound 4-[2-(4-amino-piperidin-1-yl)-5-(3-fluoro-4-methoxy-phenyl)-1-methyl-6-oxo-1,6-dihydro-pyrimidin-4-yl]-2-fluorobenzonitrile.

For research use only. We do not sell to patients.

LSD1-IN-7 Methylbenzenesulfonate Chemical Structure

LSD1-IN-7 Methylbenzenesulfonate Chemical Structure

CAS No. : 2097523-57-2

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Description

LSD1-IN-7 Methylbenzenesulfonate is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity extracted from patent WO2017079670A1, compound 4-[2-(4-amino-piperidin-1-yl)-5-(3-fluoro-4-methoxy-phenyl)-1-methyl-6-oxo-1,6-dihydro-pyrimidin-4-yl]-2-fluorobenzonitrile[1].

IC50 & Target

Lysine specific demethylase-1 (LSD1)[1]

In Vivo

LSD1-IN-7 in combination with other LSD1 inhibitor can be treatment of cancer in a mammal, including breast cancer, lung cancer, prostate cancer, glioblastoma, or leukemia[1].

Molecular Weight

623.67

Formula

C₃₁H₃₁F₂N₅O₅S

CAS No.

2097523-57-2

SMILES

N#CC1=CC=C(C(N=C(N2CCC(N)CC2)N3C)=C(C4=CC=C(OC)C(F)=C4)C3=O)C=C1F.O=S(C5=CC=C(C)C=C5)(O)=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

LSD1-IN-7Histone DemethylaseInhibitorinhibitorinhibit

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LSD1-IN-7 Methylbenzenesulfonate
Cat. No.:
HY-129388
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