NH2-c[X-R-L-S-X]-K-G-P-(D-2Nal)
NH2-c[X-R-L-S-X]-K-G-P-(D-2Nal) (compound 40), a macrocyclic analogue of Ape13, is a potent APJ agonist (Ki=5.7 nM). NH2-c[X-R-L-S-X]-K-G-P-(D-2Nal) exhibits a favorable Gα12-biased signaling and an increased in vivo half-life.
For research use only. We do not sell to patients.
- CAS No.: 2891469-81-9
- Formula: C49H73N13O11
- Molecular Weight:1020.18
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Description
IC50 & Target
APJ[1]
Chemical Information
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CAS No. 2891469-81-9
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Molecular Weight 1020.18
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Formula C49H73N13O11
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)