Orexin receptor antagonist 7
Orexin receptor antagonist 7 (Compound 34) is an antagonist of the orexin receptor (OX1R), with a Ki value of 4.05 nM. Orexin receptor antagonist 7 shows no detectable activity towards OX2R and has very low affinities for the three opioid receptors (μ, δ, κ) (Ki > 1,000 nM). Orexin receptor antagonist 7 can be used for research on opioid addiction.
For research use only. We do not sell to patients.
- CAS No.: 2096315-41-0
- Formula: C31H32N2O7S
- Molecular Weight:576.66
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All Orexin Receptor (OX Receptor) Isoforms
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Biological Activity
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OX1 Receptor 4.05 nM (Ki) |
Chemical Information
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CAS No. 2096315-41-0
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Molecular Weight 576.66
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Formula C31H32N2O7S
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SMILES
O[C@]12[C@@]34C5=C(C[C@@]2([H])N(CC4)S(=O)(C6=CC=CC=C6)=O)C=CC(OC)=C5O[C@@]3([H])[C@@H](CC1)N(C)C(/C=C/C7=COC=C7)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)