1. GPCR/G Protein
    Neuronal Signaling
  2. Dopamine Receptor
    5-HT Receptor
  3. Paliperidone palmitate

Paliperidone palmitate (Synonyms: 9-Hydroxyrisperidone palmitate)

Cat. No.: HY-A0019A Purity: 98.16%
Handling Instructions

Paliperidone palmitate (9-Hydroxyrisperidone palmitate), an atypical long-acting antipsychotic agent, is an ester prodrug of Paliperidone. Paliperidone is a dopamine antagonist and 5-HT2A antagonist of the atypical antipsychotic class. Paliperidone palmitate shows efficacy against schizophrenia.

For research use only. We do not sell to patients.

Paliperidone palmitate Chemical Structure

Paliperidone palmitate Chemical Structure

CAS No. : 199739-10-1

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 77 In-stock
Estimated Time of Arrival: December 31
10 mg USD 70 In-stock
Estimated Time of Arrival: December 31
50 mg   Get quote  
100 mg   Get quote  

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Based on 1 publication(s) in Google Scholar

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Description

Paliperidone palmitate (9-Hydroxyrisperidone palmitate), an atypical long-acting antipsychotic agent, is an ester prodrug of Paliperidone. Paliperidone is a dopamine antagonist and 5-HT2A antagonist of the atypical antipsychotic class. Paliperidone palmitate shows efficacy against schizophrenia[1].

IC50 & Target[1]

D2 Receptor

 

5-HT2A Receptor

 

Clinical Trial
Molecular Weight

664.89

Formula

C₃₉H₅₇FN₄O₄

CAS No.

199739-10-1

SMILES

O=C(OC1CCCN(C1=NC(C)=C2CCN3CCC(C4=NOC5=C4C=CC(F)=C5)CC3)C2=O)CCCCCCCCCCCCCCC

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

4°C, sealed storage, away from moisture and light

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)

Solvent & Solubility
In Vitro: 

Ethanol : 2 mg/mL (3.01 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 1.5040 mL 7.5200 mL 15.0401 mL
5 mM --- --- ---
10 mM --- --- ---
*Please refer to the solubility information to select the appropriate solvent.
References
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Keywords:

Paliperidone9-HydroxyrisperidoneDopamine Receptor5-HT ReceptorSerotonin Receptor5-hydroxytryptamine Receptorantipsychoticesterprodrugschizophreniaatypicallong-actingInhibitorinhibitorinhibit

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Product Name:
Paliperidone palmitate
Cat. No.:
HY-A0019A
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