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Cat. No.: HY-A0019AS

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Paliperidone palmitate-d₄

(Synonyms: 9-Hydroxyrisperidone palmitate-d₄)

Paliperidone palmitate-d₄ (9-Hydroxyrisperidone palmitate-d₄) is the deuterium labeled Paliperidone palmitate (HY-A0019A). Paliperidone palmitate is an orally effective competitive antagonist of dopamine D2 receptors and 5-hydroxytryptamine 2A (5-HT2A) receptors that can cross the blood-brain barrier. Paliperidone palmitate competitively inhibits the effects of dopamine and 5-hydroxytryptamine by binding to dopamine D2 receptors and 5-HT2A receptors, regulating the balance of the neurotransmitter system and thus exerting antipsychotic activity. Paliperidone palmitate is mainly used in the research field of schizophrenia.

For research use only. We do not sell to patients.

CAS No.: 1794685-21-4
Formula: C₃₉H₅₃D₄FN₄O₄
Molecular Weight:668.92

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (237 KB)

Paliperidone palmitate-d₄ Chemical Structure

CAS No.: 1794685-21-4

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Biological Activity
- Description
- In Vitro
- Application
Chemical Information
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Biological Activity

Description

All 5-HT Receptor Isoforms :

All Dopamine Receptor Isoforms :

In Vitro

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Application

1. This compound can be used as a tracer
2. This compound can be used as an internal standard for quantitative analysis by NMR, GC-MS, or LC-MS.

Chemical Information

CAS No. 1794685-21-4
Unlabeled Cas 199739-10-1
Molecular Weight 668.92
Formula C₃₉H₅₃D₄FN₄O₄
SMILES

FC1=CC=C(C(C2CCN(CC2)C([2H])([2H])C([2H])([2H])C3=C(C)N=C(C(CCC4)OC(CCCCCCCCCCCCCCC)=O)N4C3=O)=NO5)C5=C1
Synonyms

9-Hydroxyrisperidone palmitate-d₄
Shipping

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Storage

Please store the product under the recommended conditions in the Certificate of Analysis.