Protease-Activated Receptor-1 antagonist 3
Protease-Activated Receptor-1 antagonist 3 is a potent protease-activated receptor-1 antagonist with an IC50 value of 7 nM. Protease-Activated Receptor-1 antagonist 3 shows binding affinity for hERG K+ channel with an IC50 value of 9 µM.
For research use only. We do not sell to patients.
- Formula: C30H34N4O3
- Molecular Weight:498.62
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
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Animal Model:Rats[1]
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Dosage:3 mg/kg
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Administration:I.v.
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Result:Exhibited relatively high unbound clearance values with CLu of 742 mL/min/kg, and Vd of 1.2 L/kg in rats.
Chemical Information
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Molecular Weight 498.62
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Formula C30H34N4O3
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SMILES
[H][C@]12[C@H]([C@@H]([C@@H](C)[C@H]3[C@]1(C(O[C@@H]2C)=O)CN(C(NCC)=O)C3)C)/C=C/C4=CC=C(C=N4)C5=CC=CC=C5C#N
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Protease-Activated Receptor-1 antagonist 3 Related Classifications
HY-143315 Related Classifications
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