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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
26 Results for "
Choline acetyltransferase
" in MedChemExpress (MCE) Product Catalog:
Products (26)
26 Results for "Choline acetyltransferase" in MCE Product Catalog:
13
13 Publications Verification
Research Areas:
α-NETA is a potent and noncompetitive choline acetyltransferase (ChA) inhibitor with an IC50 of 9 μM. α-NETA is a potent ALDH1A1 (IC50=0.04 µM) and chemokine-like receptor-1 (CMKLR1) antagonist. α-NETA weakly inhibits cholinesterase (ChE; IC50=84 µM) and acetylcholinesterase (AChE; IC50=300 µM). α-NETA has anti-cancer activity .
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Category:
Apocynaceae Flavonols Flavonoids Other Diseases Phenols Polyphenols Plants Apocynum venetum Linn. Disease Research Fields
Target:
3
3 Cited Publications
Cat. No.: HY-B1337S1
CAS No.: 61037-86-3
1
1 Cited Publications
Cat. No.: HY-B1337S
CAS No.: 285979-70-6
1
1 Cited Publications
Cat. No.: HY-B1337S4
Cat. No.: HY-N8376
CAS No.: 20725-03-5
Synonyms: (±)-Fustin; 3,7,3',4'-Tetrahydroxyflavanone
Category:
Target:
Cat. No.: HY-B1337S3
CAS No.: 352438-97-2
Cat. No.: HY-N4119
CAS No.: 13241-32-2
Category:
other families Flavonoids Flavonones Phenols Polyphenols Plants
Cat. No.: HY-W100403
CAS No.: 55357-38-5
Synonyms: Choline p-toluenesulfonate
Cat. No.: HY-159904
Target:
Research Areas:
ChAT IN-1 is a selective Choline Acetyltransferase (ChAT) inhibitor. It can be used to study mechanisms related to the overexpression of non-neuronal ChAT in cancers (e.g., colorectal and lung cancers) and Alzheimer’s disease (AD) .
Cat. No.: HY-N0801
CAS No.: 22338-71-2
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Target:
Research Areas:
β-NETA is a potent and noncompetitive choline acetyltransferase (ChA; IC50=76 μM) and cholinesterase (ChE; IC50=40 μM) inhibitor. β-NETA weakly inhibits acetylcholinesterase (AChE; IC50=1 mM) .
Cat. No.: HY-W127668
CAS No.: 5957-17-5
Cat. No.: HY-124892A
CAS No.: 103994-00-9
Synonyms: Acetyl-AF64
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Research Areas:
Acetylethylcholine mustard hydrochloride (Acetyl-AF64) is an inhibitor of choline acetyl-transferase that reduces the contraction frequency of the myotubes by inhibiting the synthesis of acetylethylcholine (Ach) with the half-maximal inhibitory concentration (IC50) of 1.22 mM. Acetylethylcholine mustard hydrochloride is an irreversible ligand for the high affinity choline transport system. Acetylethylcholine mustard hydrochloride is also a cholinotoxin. Acetylethylcholine mustard hydrochloride is a precursor for ethylcholine mustard aziridinium ion .
Cat. No.: HY-138199S
CAS No.: 2740875-18-5
Research Areas:
Omeprazole sulfone N-Oxide- 13C,d3 is the 13C,d3 Omeprazole sulfone N-Oxide (HY-138199). Omeprazole sulfone N-Oxide is an Omeprazole (HY-B0113) analog with binding affinity to Nilaparvata lugens choline acetyltransferase (ChAT) .
Cat. No.: HY-11055
CAS No.: 393856-87-6
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KP 544 is a potent neurotrophic protein enhancer that amplifies nerve growth factor (NGF)-induced neurite outgrowth of PC12 cells and SH-SY5Y neuroblastoma cells. KP544 also enhances choline acetyltransferase activity. KP 544 selectively interact in the differentiation pathway downstream of MAPK in a manner that amplifies nerve growth factor and cyclic AMP effects and is also neuroprotective .
Cat. No.: HY-138199S1
CAS No.: 2748468-58-6
Research Areas:
Omeprazole sulfone N-Oxide-d3 is the d3-labeled Omeprazole sulfone N-Oxide (HY-138199). Omeprazole sulfone N-Oxide is an Omeprazole (HY-B0113) analog with binding affinity to Nilaparvata lugens choline acetyltransferase (ChAT) .
Cat. No.: HY-B1337S2
CAS No.: 3035513-80-2
Cat. No.: HY-U00114
CAS No.: 324077-62-5
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Research Areas:
ZSET-845 is a cognitive enhancer which enhances choline acetyltransferase activity in the hippocampus in the rat.
Cat. No.: HY-138199
CAS No.: 158812-85-2
Target:
Research Areas:
Omeprazole sulfone N-Oxide is an Omeprazole (HY-B0113) analog with binding affinity to Nilaparvata lugens choline acetyltransferase (ChAT) .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
