2 Results for "

glial transporters

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "glial transporters" in MCE Product Catalog:

3
3 Cited Publications
Cat. No.: HY-107521
CAS No.: 480439-73-4
Purity:  99.28%
Synonyms: CF3-Bza-TBOA
Target:  

EAAT

Research Areas:  

Neurological Disease

TFB-TBOA (CF3-Bza-TBOA) is a potent glutamate transporter blocker that potently suppresses the activity of glial transporters. TFB-TBOA shows IC50 values of 22, 17, and 300 nM for glutamate transporters EAAT1, EAAT2, and EAAT3 respectively in an uptake assay using cells transiently expressing EAATs .
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Cat. No.: HY-100838
CAS No.: 117857-95-1
Synonyms: L-CCG III
Target:  

EAAT

Research Areas:  

Neurological Disease

cis-α-(Carboxycyclopropyl)glycine (L-CCG III) is a potent, competitive glutamate uptake inhibitor. cis-α-(Carboxycyclopropyl)glycine is a substrate of glutamate transporters (GluT) (EC50: 13 μM, 2 μM for EAAT 1 and EAAT 2, respectively). cis-α-(Carboxycyclopropyl)glycine inhibits a Na +-dependent high-affinity L-glutamate uptake in glial plasmalemmal vesicles (GPV) and synaptosomes .
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