2. Neuronal Signaling
  3. Sigma Receptor
  4. Trifluperidol hydrochloride

Trifluperidol hydrochloride  (Synonyms: R 2498)

Cat. No.: HY-124462 Purity: 99.4%
COA
SDS
Handling Instructions Technical Support

Trifluperidol hydrochloride is a Sigma-1 receptor antagonist with a Ki value of 3.3 nM. Trifluperidol hydrochloride is used in the study of psychosis.

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Trifluperidol hydrochloride

Trifluperidol hydrochloride 화학구조

CAS No. : 2062-77-3

사이즈 가격 재고 수량
5 mg 해외재고보유
10 mg   견적 받기  
50 mg   견적 받기  

* 장바구니에 담기 전 물품의 수량을 선택해 주십시오.

This product is a controlled substance and not for sale in your territory.

Trifluperidol hydrochloride Related Antibodies

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제품 설명

Trifluperidol hydrochloride is a Sigma-1 receptor antagonist with a Ki value of 3.3 nM. Trifluperidol hydrochloride is used in the study of psychosis[1].

분자량

445.88

화학식

C22H24ClF4NO2
CAS No.
Appearance

Solid

Color

White to off-white

SMILES

O=C(CCCN1CCC(O)(CC1)C2=CC=CC(C(F)(F)F)=C2)C3=CC=C(C=C3)F.[H]Cl
선적

Room temperature in continental US; may vary elsewhere.
보관

-20°C, sealed storage, away from moisture

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

용액&용해도
In Vitro: 

DMSO : 40 mg/mL (89.71 mM; Need ultrasonic and warming; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.2428 mL 11.2138 mL 22.4276 mL
5 mM 0.4486 mL 2.2428 mL 4.4855 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

  • 몰농도 계산기

  • 농도 희석 계산기

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass
=
Concentration
×
Volume
×
Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start)

C1

×
Volume (start)

V1

=
Concentration (final)

C2

×
Volume (final)

V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

Dosage

mg/kg

Animal weight
(per animal)

g

Dosing volume
(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
순도&문서

Purity: 99.4%

SDS (479 KB)

COA (245 KB)

Handling Instructions (2659 KB)
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.2428 mL 11.2138 mL 22.4276 mL 56.0689 mL
5 mM 0.4486 mL 2.2428 mL 4.4855 mL 11.2138 mL
10 mM 0.2243 mL 1.1214 mL 2.2428 mL 5.6069 mL
15 mM 0.1495 mL 0.7476 mL 1.4952 mL 3.7379 mL
20 mM 0.1121 mL 0.5607 mL 1.1214 mL 2.8034 mL
25 mM 0.0897 mL 0.4486 mL 0.8971 mL 2.2428 mL
30 mM 0.0748 mL 0.3738 mL 0.7476 mL 1.8690 mL
40 mM 0.0561 mL 0.2803 mL 0.5607 mL 1.4017 mL
50 mM 0.0449 mL 0.2243 mL 0.4486 mL 1.1214 mL
60 mM 0.0374 mL 0.1869 mL 0.3738 mL 0.9345 mL
80 mM 0.0280 mL 0.1402 mL 0.2803 mL 0.7009 mL
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Trifluperidol hydrochloride Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Trifluperidol2062-77-3R 2498R2498R-2498Sigma ReceptorSigma-1 receptorAntagonistantipsychoticInhibitorinhibitorinhibit

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상품명:
Trifluperidol hydrochloride
Cat. No.:
HY-124462
수량:
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SAFETY DATA SHEET (SDS)

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