GABA Receptor
Gamma-aminobutyric acid Receptor; γ-Aminobutyric acid Receptor
GABA receptors are a class of receptors that respond to the neurotransmitter gamma-aminobutyric acid (GABA), the chief inhibitory neurotransmitter in the vertebrate central nervous system. There are two classes of GABA receptors: GABAA and GABAB. GABAA receptors are ligand-gated ion channels (also known as ionotropic receptors), whereas GABAB receptors are G protein-coupled receptors (also known asmetabotropic receptors). It has long been recognized that the fast response of neurons to GABA that is blocked by bicuculline and picrotoxin is due to direct activation of an anion channel. This channel was subsequently termed the GABAA receptor. Fast-responding GABA receptors are members of family of Cys-loop ligand-gated ion channels. A slow response to GABA is mediated by GABAB receptors, originally defined on the basis of pharmacological properties.
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GABA Receptor Inhibitors
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GABA Receptor Agonists
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GABA Receptor Antagonists
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GABA Receptor Activators
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GABA Receptor Ligands
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GABA Receptor Related Products (787)
Related Products (787)
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Antibodies (14)
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Related Compound Screening Libraries (1)
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3-Methoxyphenol-d3
0 ImagesCat. No.: HY-Y1840SCAS No.: 104714-88-73-Methoxyphenol-d3 is the d3-labeled 3-Methoxyphenol (HY-Y1840). 3-Methoxyphenol is an environmental pollutant. 3-Methoxyphenol occurs in the aroma components of dried bonito. 3-Methoxyphenol potentially enhances GABA-evoked responses of α1β1 GABAA receptors by increasing the affinity of GABA binding sites. 3-Methoxyphenol is used as a flavoring substance in food and animal feed. 3-Methoxyphenol prolongs pentobarbital-induced sleeping time and reduces elevated plus maze behavior.
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epi-Aszonalenin A
0 ImagesCat. No.: HY-135154CAS No.: 908853-14-5epi-Aszonalenin A is a benzodiazepine fungal metabolite originally isolated from Aspergillus novofumigatus. epi-Aszonalenin A can be used as a psychoactive agent.
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Carburazepam
0 ImagesCat. No.: HY-U00241CAS No.: 59009-93-7Synonyms: RGH 3331; UxepamCarburazepam is a agent which derives from benzodiazepine. Benzodiazepines (BZD, BZs) are a class of psychoactive agents whose core chemical structure is the fusion of a benzene ring and a diazepine ring.
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Suclofenide
0 ImagesCat. No.: HY-U00102CAS No.: 30279-49-3Synonyms: Neosulfalepsine; PB385Suclofenide (Neosulfalepsine; PB385) is an anticonvulsant that affects GABA metabolism.
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CGP11952
0 ImagesCat. No.: HY-U00192CAS No.: 64078-09-7CGP11952 is a triazolyl-Benzaphenon resembling the benzodiazepines in its pharmacological action. CGP11952 is an experimental benzodiazepine derivative.
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Ro 41-3290
0 ImagesCat. No.: HY-U00215CAS No.: 143943-72-0Ro 41-3290 is the desethylated derivative of Ro 41-3696, which is a nonbenzodiazepine partial agonist at the benzodiazepine receptor.
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FG8119
0 ImagesCat. No.: HY-U00233CAS No.: 106447-61-4Synonyms: NNC13-8119FG8119 is a novel benzodiazepine agonist extracted from patent US 4745112 A.
