GRL018-21
Based on 1 Customer Validation
GRL018-21 is a potent and highly selective G protein-coupled receptor kinase 5 (GRK5) inhibitor with an IC50 value of 10 nM.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- 純度: 96.91%
- CAS 番号: 3061801-07-5
- 分子式: C30H25FN4O5
- 分子量:540.54
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保管条件:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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生物活性
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化学情報
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溶剤 & 溶解度
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
生物活性
化学情報
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CAS 番号 3061801-07-5
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性状 Solid
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分子量 540.54
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分子式 C30H25FN4O5
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Color Orange to red
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SMILES
FC1=CC=C([C@@H](C)NC(C2=CC=C(NC(/C3=C\C4=C(C)C(NC(C(C5=CC=CO5)=O)=O)=C(C)N4)=O)C3=C2)=O)C=C1
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
溶剤 & 溶解度
DMSO : 35 mg/mL (64.75 mM; ultrasonic and warming and heat to 60°C; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
純度とドキュメンテーション
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データシート (268 KB)
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SDS (252 KB)
- English - EN (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Korean - KR (252 KB)
- Portuguese - PT (252 KB)
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取扱説明書 (2659 KB)
参考文献
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 1.8500 mL | 9.2500 mL | 18.5000 mL | 46.2500 mL |
| 5 mM | 0.3700 mL | 1.8500 mL | 3.7000 mL | 9.2500 mL | |
| 10 mM | 0.1850 mL | 0.9250 mL | 1.8500 mL | 4.6250 mL | |
| 15 mM | 0.1233 mL | 0.6167 mL | 1.2333 mL | 3.0833 mL | |
| 20 mM | 0.0925 mL | 0.4625 mL | 0.9250 mL | 2.3125 mL | |
| 25 mM | 0.0740 mL | 0.3700 mL | 0.7400 mL | 1.8500 mL | |
| 30 mM | 0.0617 mL | 0.3083 mL | 0.6167 mL | 1.5417 mL | |
| 40 mM | 0.0463 mL | 0.2313 mL | 0.4625 mL | 1.1563 mL | |
| 50 mM | 0.0370 mL | 0.1850 mL | 0.3700 mL | 0.9250 mL | |
| 60 mM | 0.0308 mL | 0.1542 mL | 0.3083 mL | 0.7708 mL |
GRL018-21 関連分類
HY-149720 関連分類
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