1. PROTAC
  2. Target Protein Ligand-Linker Conjugate
  3. K-Ras ligand-Linker Conjugate 3

K-Ras ligand-Linker Conjugate 3 

Cat. No.: HY-130707
Handling Instructions

K-Ras ligand-Linker Conjugate 3 (Compound 001371) incorporates a ligand for FAK (a KRas recruiting moiety), and a PROTAC linker, which recruit E3 ligases (such as VHL, CRBN, MDM2, and IAP). K-Ras ligand-Linker Conjugate 3 can be extensively used for PROTAC-mediated protein degradation.

For research use only. We do not sell to patients.

K-Ras ligand-Linker Conjugate 3 Chemical Structure

K-Ras ligand-Linker Conjugate 3 Chemical Structure

CAS No. : 2378261-87-9

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 2650 In-stock
Estimated Time of Arrival: December 31
1 mg USD 550 In-stock
Estimated Time of Arrival: December 31
5 mg USD 1650 In-stock
Estimated Time of Arrival: December 31
10 mg USD 2550 In-stock
Estimated Time of Arrival: December 31
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Based on 1 publication(s) in Google Scholar

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Description

K-Ras ligand-Linker Conjugate 3 (Compound 001371) incorporates a ligand for FAK (a KRas recruiting moiety), and a PROTAC linker, which recruit E3 ligases (such as VHL, CRBN, MDM2, and IAP). K-Ras ligand-Linker Conjugate 3 can be extensively used for PROTAC-mediated protein degradation[1].

Molecular Weight

944.15

Formula

C₄₉H₆₅N₇O₁₀S

CAS No.

2378261-87-9

SMILES

O=C(N1[[email protected]@H](CC#N)CN(C2=C3C(CN(C4=C5C=CC=CC5=CC=C4)CC3)=NC(OC[[email protected]]6N(C)C[[email protected]](OCCOCCOCCOCCOS(=O)(C7=CC=C(C)C=C7)=O)C6)=N2)CC1)OC(C)(C)C

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Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

K-Ras ligand-Linker Conjugate 3Target Protein Ligand-Linker ConjugateInhibitorinhibitorinhibit

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K-Ras ligand-Linker Conjugate 3
Cat. No.:
HY-130707
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