PFI-7-O-C4-piperazin

PFI-7-O-C4-piperazin is a E3 ligase ligand-linker conjugate that can be used for synthesis of PROTACs, such as NEP162 (HY-174996). The E3 ligase ligand (PFI-7) of NEP162 is a highly selective antagonist of GID4 (KD = 0.22 μM). NEP162 is a BRD4 PROTAC degrader with anti-tumor activity[1].

For research use only. We do not sell to patients.

  • Formula: C31H41N7O2
  • Molecular Weight:543.70
  • Storage:

    Please store the product under the recommended conditions in the Certificate of Analysis.

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All E3 Ligase Ligand-Linker Conjugates Isoforms

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