(S)-Human enteropeptidase-IN-1
(S)-Human enteropeptidase-IN-1 (Compound 6c) is an orally active enteropeptidase inhibitor with low systemic exposure (IC50 (initial): 26 nM; IC50 (app): 1.8 nM). (S)-Human enteropeptidase-IN-1 promotes increased fecal protein output and effectively reduces body weight in a diet-induced obese (DIO) rat model. (S)-Human enteropeptidase-IN-1 inhibits enteropeptidase via a reversible covalent mechanism and prolongs the enzyme inactivation time. (S)-Human enteropeptidase-IN-1 can be used in anti-obesity research.
For research use only. We do not sell to patients.
- CAS No.: 1802891-23-1
- Formula: C20H18N4O7
- Molecular Weight:426.38
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
-
Biological Activity
-
Chemical Information
- Purity & Documentation
- References
-
Help & FAQs
Biological Activity
Chemical Information
-
CAS No. 1802891-23-1
-
Molecular Weight 426.38
-
Formula C20H18N4O7
-
SMILES
O=C([C@@]1(CC(O)=O)CC(C2=CC=CC(OC(C3=CC=C(NC(N)=N)C=C3)=O)=C2)=NO1)O
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
(S)-Human enteropeptidase-IN-1 Related Classifications
HY-147927A Related Classifications
Powered by Bioz