88 Results for "

G-{d-Arg}-GDSPASSK

" in MedChemExpress (MCE) Product Catalog:
Products (88)

88 Results for "G-{d-Arg}-GDSPASSK" in MCE Product Catalog:

Cat. No.: HY-P7061
CAS No.: 143413-49-4
Research Areas:  

Infection Endocrinology

ALX 40-4C is a small peptide inhibitor of the chemokine receptor CXCR4, inhibits SDF-1 from binding CXCR4 with a Ki of 1 μM, and suppresses the replication of X4 strains of HIV-1; ALX 40-4C Trifluoroacetate also acts as an antagonist of the APJ receptor, with an IC50 of 2.9 μM.
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Cat. No.: HY-P10644
CAS No.: 1831064-63-1
Target:  

Fluorescent Dye

Research Areas:  

Cancer

CPP9 is a small, amphipathic, cyclic cell penetrating peptide (CPP). CPPs bind directly to the plasma membrane phospholipids and enter mammalian cells via endocytosis, followed by efficient release from the endosome. CPP9 can be used for intracellular delivery of therapeutic agents and chemical probes .
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Cat. No.: HY-P4474A
Target:  

Inhibitory Antibodies

Research Areas:  

Others

Pz-Pro-Leu-Gly-Pro-d-Arg TFA is a synthetic polypeptide substrate. Pz-Pro-Leu-Gly-Pro-d-Arg TFA can be used to detect the collagenase-like activity of enzymes from various sources, such as Bacillus sp. AH-101 .
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Cat. No.: HY-P3582A
Target:  

GnRH Receptor

Research Areas:  

Endocrinology

sGnRH-A acetate is a salmon gonadotropin-releasing hormone (GnRH) analogue. sGnRH-A acetate stimulates growth hormone secretion. sGnRH-A acetate also can be used as an inducer of ovulation by artificial insemination .
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Cat. No.: HY-P10923
CAS No.: 592544-81-5
Target:  

Cathepsin

Research Areas:  

Others

KYS-1 is a selective substrate for cathepsin E with a Km value of 1.9 μM. KYS-1 was incubated with cathepsin E (1.0 ng) with the pH optimum of approximately pH 4.0 .
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Cat. No.: HY-P2498
CAS No.: 839730-93-7
Target:  

Cathepsin

Research Areas:  

Others

Cathepsin D and E FRET Substrate is a fluorogenic substrate for cathepsins D and E and not for B, H or L. The cleavage occurs at the Phe-Phe amide bond resul. Cathepsin D and E FRET Substrate is a valuable tool for routine assays and for mechanistic studies on cathepsins E and D .
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Cat. No.: HY-P5518A
[Des-Arg10]-HOE I40 TFA is a potent bradykinin B1 receptor antagonist .
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Cat. No.: HY-P3880
CAS No.: 84676-91-5
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

(D-Arg1,D-Pro2,D-Trp7,9,L-Leu11)-Substance P is a neuropeptide Substance P (HY-P0201) antagonist .
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Cat. No.: HY-P3881
CAS No.: 115760-58-2
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

(D-Arg1,D-Pro2,D-Phe7,D-His9)-Substance P is a selective NK1 receptor antagonist .
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Cat. No.: HY-P11374
Target:  

Bcl-2 Family Apoptosis

Research Areas:  

Cancer

Bid BH3-Gly-r8 is Bid BH3 linked to eight arginine residues. Bid BH3-Gly-r8 shows no difference in apoptotic effects compared to its unmodified peptide homologue. Bid BH3 has high affinity for Bax and Bcl-2. Bid BH3-Gly-r8 can be used in the research of tumors .
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Cat. No.: HY-P10331
CAS No.: 2757292-12-7
Target:  

SDCBP

Research Areas:  

Cancer

KSL 128114, a peptide inhibitor of syntenin, binds the PDZ1 domain of syntenin with nanomolar affinity. KSL 128114 is resistant toward degradation in human plasma and mouse hepatic microsomes and displays a global PDZ domain selectivity for syntenin .
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Cat. No.: HY-P5131
CAS No.: 255861-98-4
Target:  

Opioid Receptor

Research Areas:  

Others

[Dmt1]DALDA is a potent and long-acting analgesic binds to the mu opioid receptor with high affinity and selectivity. [Dmt1]DALDA is a full agonist at hMOR (Kd = 0.199 nM) and hDOR, but only partial agonist against hKOR .
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Cat. No.: HY-P4750
CAS No.: 93942-91-7
Target:  

GHSR

Research Areas:  

Endocrinology

Acetyl-(D-Arg2)-GRF (1-29) amide (human) is an antagonist of growth hormone releasing factor (GRF). Acetyl-(D-Arg2)-GRF (1-29) amide (human) inhibits the release of growth hormone (GH) and can be used for endocrine research .
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Cat. No.: HY-P10918
Target:  

Inhibitory Antibodies

Research Areas:  

Inflammation/Immunology

F11R peptide TFA is a F11 receptor molecule. F11R peptide TFA inhibits anti-F11R antibody-induced platelet aggregation, and inhibits the adhesion of platelets to cytokine (TNFα and INF-γ)-inflammed endothelial cells. F11R peptide TFA can be used for research of atherosclerotic plaques and associated thrombotic disease .
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Cat. No.: HY-P10790
CAS No.: 1332850-08-4
Target:  

Microtubule/Tubulin

Research Areas:  

Cancer

Breast cancer targeting peptide 18–4 is a KRT1 receptor-targeting peptide, with a Kd of 0.98 μM. The amino acid sequence of Breast cancer targeting peptide 18–4 is WxEAAYQrFL, and it is an analogue of P160 peptide (HY-P10789). When covalently conjugated with the anticancer peptide MccJ25, Breast cancer targeting peptide 18–4 significantly increases the cellular uptake of MccJ25 in breast cancer cells and enhances its anticancer activity. The covalent conjugate exhibits IC50 values of 14.2, 20, and 25 μM against MCF-7, MDA-MB-435, and MDA-MB-435-MDR cells, respectively .
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Cat. No.: HY-P10394
CAS No.: 2376306-14-6
DP32 is a bifunctional compound that contains an opioid receptor (MOP) agonist and a neuropeptide FF receptor (NPFFR) antagonist. DP32 can be used in analgesia-related research .
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Cat. No.: HY-P5010
CAS No.: 745816-74-4
Target:  

Vasopressin Receptor

Research Areas:  

Cardiovascular Disease

(D-Arg8)-Inotocin is a potent, selective and competitive antagonist of vasopressin receptor (V1aR), with a Ki of 1.3 nM. (D-Arg8)-Inotocin shows more than 3000-fold selectivity for the human V1aR over the other three subtypes, OTR, V1bR and V2R .
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Cat. No.: HY-P3397
CAS No.: 221377-79-3
Target:  

GHR

Research Areas:  

Cancer

JV-1-36 is a growth hormone-releasing hormone (GHRH) antagonist. JV-1-36 inhibits the production of reactive oxygen species in A549 lung cancer cells. JV-1-36 can be used to study the effect of GHRH antagonists in vitro .
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Cat. No.: HY-P10118A
Target:  

Cathepsin

Research Areas:  

Others

Cathepsin L-IN-3 (Compound cat L inh. 7) TFA is selective a noncovalent cathepsin L inhibitor with a Ki of 4.3 nM .
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Cat. No.: HY-P11405
CAS No.: 122481-75-8
Target:  

Neurotensin Receptor

Research Areas:  

Neurological Disease Cancer

[D-Arg1, D-Trp5, 7, 9, Leu11]-Substance P is a potent inhibitor of cell growth in small cell lung cancer (SCLC). [D-Arg1, D-Trp5, 7, 9, Leu11]-Substance P is also a neuropeptide antagonist, capable of blocking colony formation stimulated by various neuropeptides (including vasopressin and bradykinin). [D-Arg1, D-Trp5, 7, 9, Leu11]-Substance P inhibits the mobilization of Ca 2+ and the activation of mitogen-activated protein kinases induced by vasopressin or bradykinin. [D-Arg1, D-Trp5, 7, 9, Leu11]-Substance P inhibits the growth of H-69 xenograft tumors in nude mice .
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