(D-Arg8)-Inotocin
(D-Arg8)-Inotocin is a potent, selective and competitive antagonist of vasopressin receptor (V1aR), with a Ki of 1.3 nM. (D-Arg8)-Inotocin shows more than 3000-fold selectivity for the human V1aR over the other three subtypes, OTR, V1bR and V2R.
For research use only. We do not sell to patients.
- CAS No.: 745816-74-4
- Formula: C39H68N14O11S2
- Molecular Weight:973.17
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All Vasopressin Receptor Isoforms
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Biological Activity
Chemical Information
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CAS No. 745816-74-4
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Molecular Weight 973.17
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Formula C39H68N14O11S2
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Sequence
Cys-Leu-Ile-Thr-Asn-Cys-Pro-{d-Arg}-Gly-NH2 (Disulfide bridge: Cys1-Cys6)
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Sequence Shortening
CLITNCP-{d-Arg}-G-NH2 (Disulfide bridge: Cys1-Cys6)
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)