92 Results for "

OPCs

" in MedChemExpress (MCE) Product Catalog:
Products (92)

92 Results for "OPCs" in MCE Product Catalog:

Cat. No.: HY-17464S2
CAS No.: 1073608-03-3
Synonyms: OPC 13013-d2
Cilostazol-d2 (OPC 13013-d2) is deuterium labeled Cilostazol. Cilostazol (OPC 13013) is a potent and selective inhibitor of phosphodiesterase (PDE) 3A, the isoform of PDE 3 in the cardiovascular system, with an IC50 of 0.2 μM .
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Cat. No.: HY-106781A
CAS No.: 1329509-60-5
Purity:  98.99%
Target:  

Dopamine Receptor

Research Areas:  

Neurological Disease

OPC 4392 hydrochloride is an agonist for presynaptic dopamine receptor and an antagonist for postsynaptic D2 receptor. OPC 4392 reverses the Reserpine (HY-N0480)-induced dopamine accumulation, inhibits Apomorphine (HY-12723)-induced stereotypic and climbing behaviors in mouse models .
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Cat. No.: HY-100665S
CAS No.: 2749328-53-6
Synonyms: OPC-14857-d8; DM-14857-d8
Dehydroaripiprazole-d8 is deuterium labeled Dehydroaripiprazole. Dehydroaripiprazole (OPC-14857) is an active metabolite of Aripiprazole. Aripiprazole is an antipsychotic agent and is metabolized by CYP3A4 and CYP2D6 forming mainly Dehydroaripiprazole. Dehydroaripiprazole has with antipsychotic activity equivalent to Aripiprazole .
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Cat. No.: HY-117488
CAS No.: 146761-69-5
Synonyms: (S)-OPC-17116; (S)-dl-Grepafloxacin
Target:  

Bacterial

Research Areas:  

Infection

(S)-Grepafloxacin ((S)-OPC-17116) is the S-enantiomer of Grepafloxacin (HY-A0147) .
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Cat. No.: HY-135910R
CAS No.: 73963-62-9
Synonyms: OPC-13015 (Standard)
3,4-Dehydro Cilostazol (Standard) is the analytical standard of 3,4-Dehydro Cilostazol. This product is intended for research and analytical applications. 3,4-Dehydro Cilostazol (OPC-13015) is an active metabolite of Cilostazol (CLZ; HY-17464). 3,4-Dehydro Cilostazol is used for pharmacokinetic study .
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Cat. No.: HY-135910S
CAS No.: 1073608-13-5
Synonyms: OPC-13015-d11
3,4-Dehydro Cilostazol-d11 is deuterated labeled 3,4-Dehydro Cilostazol (HY-135910). 3,4-Dehydro Cilostazol (OPC-13015) is an active metabolite of Cilostazol (CLZ; HY-17464). 3,4-Dehydro Cilostazol is used for pharmacokinetic study .
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Cat. No.: HY-U00194
CAS No.: 79644-90-9
Synonyms: Flumenique; OPC7241; DM8966
Target:  

Bacterial

Research Areas:  

Infection

Vebufloxacin (Flumenique; OPC7241; DM8966) exhibits potent antibacterial activity against gram-positive and -negative bacteria.
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Cat. No.: HY-B0506S1
Synonyms: OPC7251-d5
Nadifloxacin-d5 (OPC7251-d5) is deuterium labeled Nadifloxacin (HY-B0506). Nadifloxacin (OPC7251) is a broad-spectrum quinolone antibiotic. Nadifloxacin inhibits bacterial DNA gyrase and topoisomerase IV, interfering with DNA replication. It also suppresses the production of proinflammatory cytokines (such as IL-1α, IL-6, and IL-8). Nadifloxacin exhibits antibacterial activity against various pathogens, including Propionibacterium acnes and Staphylococcus aureus. Nadifloxacin also exhibits anti-inflammatory activity. Nadifloxacin can be used in the research of skin infections such as acne vulgaris, folliculitis, and impetigo .
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Cat. No.: HY-134082A
CAS No.: 84601-19-4
Target:  

Phospholipase

Research Areas:  

Inflammation/Immunology

(Z)-Oleyloxyethyl phosphorylcholine ((Z)-OPC) is an isomer of Oleyloxyethyl phosphorylcholine (OPC). Oleyloxyethyl phosphorylcholine is an inhibitor of secreted Phospholipase A2 (sPLA2), which is involved in the biosynthesis of proinflammatory lipid media. Oleyloxyethyl phosphorylcholine can be used to study inflammatory diseases. Oleyloxyethyl phosphorylcholine also modified the red blood membrane and was used to bind the oxygen-carrying liquid perfluorocarbons as an antivenom agent to reduce toxin-induced hemolysis .
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Cat. No.: HY-100665R
CAS No.: 129722-25-4
Synonyms: OPC-14857 (Standard); DM-14857 (Standard)
Research Areas:  

Neurological Disease

Dehydroaripiprazole (Standard) is the analytical standard of Dehydroaripiprazole. This product is intended for research and analytical applications. Dehydroaripiprazole (OPC-14857) is an active metabolite of Aripiprazole (HY-14546) and dopamine D2/D3 receptor partial agonist. Dehydroaripiprazole also has certain affinity for serotonin 5-HT1A, 5-HT2A and 5-HT2B receptors. Dehydroaripiprazole has antipsychotic activity equivalent to Aripiprazole .
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Cat. No.: HY-123593R
CAS No.: 138470-70-9
Synonyms: OPC-31260 hydrochloride (Standard)
Mozavaptan (hydrochloride) (Standard) is the analytical standard of Mozavaptan (hydrochloride). This product is intended for research and analytical applications. Mozavaptan hydrochloride (OPC-31260 hydrochloride) is a benzazepine derivative and a potent, selective, competitive and orally active vasopressin V2 receptor antagonist with an IC50 of 14 nM. Mozavaptan hydrochloride shows ~85-fold selectivity for V2 receptor over V1 receptor (IC50 of 1.2 μM), and can antagonize the antidiuretic action of arginine vasopressin (AVP) in vivo. Mozavaptan hydrochloride has the potential for hyponatremia, syndrome of inappropriate antidiuretic hormone (SIADH), and congestive heart failure treatment .
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Cat. No.: HY-17464S
CAS No.: 1073608-02-2
Cilostazol-d11 is the deuterium labeled Cilostazol. Cilostazol (OPC 13013) is a potent and selective inhibitor of phosphodiesterase (PDE) 3A, the isoform of PDE 3 in the cardiovascular system, with an IC50 of 0.2 μM .
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Cat. No.: HY-17464R
CAS No.: 73963-72-1
Synonyms: OPC 13013 (Standard)
Cilostazol (Standard) is the analytical standard of Cilostazol. This product is intended for research and analytical applications. Cilostazol (OPC 13013) is a potent and selective inhibitor of phosphodiesterase (PDE) 3A, the isoform of PDE 3 in the cardiovascular system, with an IC50 of 0.2 μM .
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Cat. No.: HY-126785
CAS No.: 108392-27-4
Synonyms: Colorimetric Elastase Substrate
Target:  

Elastase

Research Areas:  

Others

Suc-AAP-Abu-pNA (Colorimetric Elastase Substrate) is a specific substrate for pancreatic elastase (Km = 100 μM; Kcat/Km = 35,300 s -1 M -1 for rat pancreatic elastase; Km = 30 μM; Kcat/Km = 351,000 s -1 M -1 for porcine pancreatic elastase). Suc-AAP-Abu-pNA also promotes OPC migration .
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Cat. No.: HY-B0506R
CAS No.: 124858-35-1
Synonyms: OPC7251 (Standard)
Nadifloxacin (Standard) is the analytical standard of Nadifloxacin (HY-B0506). This product is intended for research and analytical applications. Nadifloxacin (OPC7251) is a broad-spectrum quinolone antibiotic. Nadifloxacin inhibits bacterial DNA gyrase and topoisomerase IV, interfering with DNA replication. It also suppresses the production of proinflammatory cytokines (such as IL-1α, IL-6, and IL-8). Nadifloxacin exhibits antibacterial activity against various pathogens, including Propionibacterium acnes and Staphylococcus aureus. Nadifloxacin also exhibits anti-inflammatory activity. Nadifloxacin can be used in the research of skin infections such as acne vulgaris, folliculitis, and impetigo .
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Cat. No.: HY-164961
CAS No.: 204135-86-4
OPC-8:0 is a nucleoside metabolite.
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Cat. No.: HY-106829A
CAS No.: 123941-50-4
Target:  

Others

Research Areas:  

Cardiovascular Disease

OPC 8490 is a stimulant. OPC 8490 has a positive inotropic effect. OPC 8490 can be used for research on heart failure .
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Cat. No.: HY-134940S1
Synonyms: OPC-167832-d4
Quabodepistat-d4 (OPC-167832-d4) is the deuterium labeled Quabodepistat (HY-134940). Quabodepistat (OPC-167832) is a potent and orally active dprE1 inhibitor with an IC50 of 0.258 μM. Quabodepistat has antituberculosis activity and can be used for the research of tuberculosis caused by Mycobacterium tuberculosis .
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Cat. No.: HY-CE00892
Synonyms: 3-Hydroxy-OPC4-coenzyme A
Research Areas:  

Metabolic Disease

3-Hydroxy-OPC4-CoA (3-Hydroxy-OPC4-coenzyme A) is a coenzyme A derivative.
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Cat. No.: HY-CE00895
Synonyms: 3-Hydroxy-OPC8-coenzyme A
Research Areas:  

Metabolic Disease

3-Hydroxy-OPC8-CoA (3-Hydroxy-OPC8-coenzyme A) is a coenzyme A derivative.
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