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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
3 Results for "
Akt3 degrader 1
" in MedChemExpress (MCE) Product Catalog:
Products (3)
3 Results for "Akt3 degrader 1" in MCE Product Catalog:
Target:
Research Areas:
Akt3 degrader 1 is an orally active selective Akt3 degrader with a DC50 of 13 nM. Akt3 degrader 1 binds to the PH domain of Akt3 to trigger proteasome-mediated degradation, with minimal effects on Akt1/Akt2. Akt3 degrader 1 inhibits cancer cell growth. Akt3 degrader 1 can be used for the research of non-small cell lung cancer .
Cat. No.: HY-175975
CAS No.: 3048204-93-6
PROTAC Akt3 Degrader-1 is a highly efficient and selective PROTAC degrader targeting Akt3. PROTAC Akt3 Degrader-1 shows weak antiproliferative activity in 36 cell lines. PROTAC Akt3 Degrader-1 can be used for the study of Triple-negative breast cancer and melanoma .
Cat. No.: HY-175976
CAS No.: 2794098-49-8
Research Areas:
Akt3 ligand-1 is an Akt3 inhibitor (IC50 = 0.1 nM) and a ligand for the target protein for PROTAC (Akt3). Akt3 ligand-1 can be used to synthesize PROTAC Akt3 Degrader-1(HY-175975) .
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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
