3 Results for "

human-derived liver microsomes

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "human-derived liver microsomes" in MCE Product Catalog:

Cat. No.: HY-149495
Target:  

PROTACs CDK

Research Areas:  

Cancer

CP-07 is a selective flavonoid-based PROTAC degrader that targets and degrades CDK9. CP-07 exhibits an IC50 of 3.3 nM against CDK9/cyclin T1, and induces CDK9 degradation in a concentration-dependent manner in 22RV1 cells with a DC50 of 43 nM. CP-07 rapidly triggers ligand-dependent and proteasome-dependent degradation of CDK9. CP-07 can be applied in prostate cancer-related research .
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Cat. No.: HY-N19921
CAS No.: 144608-09-3
Schizotenuin A is a and hIAPP fibrillation inhibitor with human-derived IC50 values of 2.93 µM and 0.58 µM, respectively, and exhibits antioxidant activity. Schizotenuin A scavenges DPPH free radicals and inhibits lipid peroxidation in rat liver microsomes. Schizotenuin A can be used in research related to Alzheimer's disease and type 2 diabetes .
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Cat. No.: HY-114572
CAS No.: 1635405-90-1
Target:  

c-Met/HGFR

Research Areas:  

Cancer

1D-2 is a c-Met protein kinase inhibitor, with a human-derived IC50 of 1.45 nM. 1D-2 inhibits the proliferation of cancer cells and exhibits metabolic stability in human and rat liver microsomes. 1D-2 can be used in related research on non-small cell lung cancer .
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