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GHSR Related Products (69)
Related Products (69)
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L-692585
0 ImagesL-692585 is a potent and nonpeptidyl growth hormone secretagogue receptor (GHS-R1a) agonist, with a Ki of 0.8 nM. L-692585 acts directly on somatotropes causing GH release.
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Emoghrelin
0 ImagesCat. No.: HY-N12348CAS No.: 928262-58-2Emoghrelin, isolated from? Heshouwu Polygonum multiflorum, stimulates growth hormone secretion via activation of the ghrelin receptor.
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(S)-PF-5190457
0 ImagesCat. No.: HY-12584APurity: 99.27%Synonyms: (S)-PF-05190457(S)-PF-5190457 ((S)-PF-05190457) is the S-enantiomer of PF-5190457 (HY-12584). PF-5190457 (PF-05190457) is a potent and selective ghrelin receptor inverse agonist with a pKi of 8.36.
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Acetyl-(D-Arg2)-GRF (1-29) amide (human)
0 ImagesAcetyl-(D-Arg2)-GRF (1-29) amide (human) is an antagonist of growth hormone releasing factor (GRF). Acetyl-(D-Arg2)-GRF (1-29) amide (human) inhibits the release of growth hormone (GH) and can be used for endocrine research.
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(αR,8aS)-GSK1614343
0 Images(αR,8aS)-GSK1614343 is the isomer of GSK1614343 (HY-113906). GSK1614343 is the potent antagonist of growth hormone secretagogues type 1a (GHS1a) receptors.
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GHRF, mouse TFA
0 ImagesCat. No.: HY-P3596APurity: 98.87%Synonyms: Mouse growth hormone-releasing factor TFAGHRF, mouse TFA, a mouse growth hormone-releasing factor, is a peptide containing 44 amino acids. GHRF, mouse TFA stimulates the release and synthesis of growth hormone.
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Somatostatin-25
0 ImagesCat. No.: HY-P1547CAS No.: 76461-17-1Somatostatin-25 is a endogenous neuropeptide hormone that shows inhibitory activity against secretion of growth hormone.
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L-692429
0 ImagesSynonyms: MK-0751L-692429 (MK-0751) is a benzolactam derivative and a nonpeptidyl growth hormone secretagogue (GHS) agonist. L-692429 binds to G protein-coupled receptor with a Ki of 63 nM.
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Meranzin
0 ImagesMeranzin is an orally active antidepressant and GHSR modulator. Meranzin significantly upregulates the expression levels of brain-derived neurotrophic factor and p-mTOR in the hippocampus via the ghrelin-growth hormone secretagogue receptor pathway. Meranzin regulates blood oxygen level-dependent signals in the hippocampus-thalamus-basal ganglia circuit, attenuates reward system activation, and promotes the normalization of related hormone levels. Meranzin effectively ameliorates depression-like behaviors and gastrointestinal hypomotility, and can be used in research related to depression and major depressive disorder.
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(D-Ala2)-GRF (1-29) amide (human)
0 Images(D-Ala2)-GRF (1-29) amide (human) is a superagonist of GRF, exhibiting extremely high GH-releasing activity about 50 times that of GRF (1-29) in both pigs and rats.
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Relamorelin
0 ImagesCat. No.: HY-19884CAS No.: 661472-41-9Synonyms: RM-131; BIM-28131Relamorelin (RM-131), a pentapeptide ghrelin analog, is a selective ghrelin/growth hormone secretagogue receptor (GHSR) agonist with a Ki of 0.42 nM for GHS-1a receptor. Relamorelin is centrally penetrant. Relamorelin increases growth hormone levels and accelerates gastric emptying. Relamorelin has the potential for cachexia, gastroparesis, and gastric/intestinal dysmobility disorders research.
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Relamorelin acetate
0 ImagesCat. No.: HY-19884ACAS No.: 1809080-14-5Synonyms: RM-131 acetate; BIM-28131 acetateRelamorelin (RM-131) acetate, a pentapeptide ghrelin analog, is a selective ghrelin/growth hormone secretagogue receptor (GHSR) agonist with a Ki of 0.42 nM for GHS-1a receptor. Relamorelin acetate is centrally penetrant. Relamorelin acetate increases growth hormone levels and accelerates gastric emptying. Relamorelin acetate has the potential for cachexia, gastroparesis, and gastric/intestinal dysmobility disorders research.
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Ghrelin receptor full agonist-2
0 ImagesCat. No.: HY-145364CAS No.: 2602452-73-1Ghrelin receptor full agonist-2 (compound 12j) is a highly potent Ghrelin receptor full agonist.
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GSK894490A
0 ImagesCat. No.: HY-115272CAS No.: 1012035-06-1GSK894490A is a non-peptide ghrelin receptor agonist.
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GSK1614343
0 ImagesCat. No.: HY-113906CAS No.: 1092076-04-4GSK1614343 is the potent antagonist of growth hormone secretagogues type 1a (GHS1a) receptors. GSK1614343 inhibits the calcium response induced by ghrelin with a pIC50 value of 7.90. GSK1614343 represents a useful tool to investigate the physiological relevance of the ghrelin system in rat models.
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L-739943
0 ImagesCat. No.: HY-118995CAS No.: 195248-02-3L-739943 is a potent, and orally active growth hormone (GH) secretagogue with an ED50 of 1 nM. L-739943 stimulates GH release in beagle dogs. L-739943 can be used for GH-related diseases research.
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BMS-604992 free base
0 ImagesCat. No.: HY-14495ACAS No.: 760944-56-7Synonyms: EX-1314 free baseBMS-604992 (EX-1314) free base is a selective, orally active small-molecule growth hormone secretagogue receptor (GHSR) agonist. BMS-604992 free base demonstrates high-affinity binding (ki=2.3 nM) and potent functional activity (EC50=0.4 nM). BMS-604992 free base can stimulate food intake in rodents.
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Substituted piperidines-1
0 ImagesCat. No.: HY-100305CAS No.: 170842-46-3Substituted piperidines-1 is a compound that can promote the release of growth hormone in humans and animals.
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CP-464709
0 ImagesCat. No.: HY-19454CAS No.: 193272-70-7CP-464709 is a Ghrelin receptor agonist that can penetrate the blood-brain barrier. CP-464709 causes an increase in blood pressure by activating pre sympathetic neurons in the spinal cord. CP-464709 causes biphasic blood pressure response when administered intravenously, while intrathecal administration only causes pressor. CP-464709 can be used for research on cardiovascular conditions.
