2. GPCR/G Protein
  3. GHSR
  4. (S)-PF-5190457

(S)-PF-5190457  (Synonyms: (S)-PF-05190457)

Cat. No.: HY-12584A Purity: 99.27%
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(S)-PF-5190457 ((S)-PF-05190457) is the S-enantiomer of PF-5190457 (HY-12584). PF-5190457 (PF-05190457) is a potent and selective ghrelin receptor inverse agonist with a pKi of 8.36.

For research use only. We do not sell to patients.

(S)-PF-5190457

(S)-PF-5190457 Chemical Structure

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Based on 1 publication(s) in Google Scholar

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Description

(S)-PF-5190457 ((S)-PF-05190457) is the S-enantiomer of PF-5190457 (HY-12584). PF-5190457 (PF-05190457) is a potent and selective ghrelin receptor inverse agonist with a pKi of 8.36[1].

Molecular Weight

512.67

Formula

C29H32N6OS
Appearance

Solid

Color

White to off-white

SMILES

CC1=NC=NC(C2=CC(CC[C@@H]3N4CC5(CCN(C(CC6=CN7C=C(C)SC7=N6)=O)CC5)C4)=C3C=C2)=C1
Shipping

Room temperature in continental US; may vary elsewhere.
Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
Purity & Documentation
References
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(S)-PF-5190457 Related Classifications

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The molarity calculator equation

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

(S)-PF-5190457(S)-PF-05190457GHSRGrowth hormone secretagogue receptorGhrelin receptorS-enantiomer of PF-5190457ghrelin receptorInhibitorinhibitorinhibit

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