CysLT1 receptor antagonist-1
CysLT1 receptor antagonist-1 (Compound 4) is an antagonist for cysteinyl leukotriene receptor 1 (CysLT1R) with an IC50 of 3.9 μM. CysLT1 receptor antagonist-1 exhibits weak agonist activity against G-protein-coupled bile acid receptor 1 (GPBAR1) with an efficact of 23% at 10 μM. CysLT1 receptor antagonist-1 can be used for asthma and allergic diseases researchs.
For research use only. We do not sell to patients.
- CAS No.: 119515-00-3
- Formula: C18H15NO3
- Molecular Weight:293.32
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
All Leukotriene Receptor Isoforms
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Biological Activity
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CysLT1 3.9 μM (IC50) |
Chemical Information
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CAS No. 119515-00-3
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Molecular Weight 293.32
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Formula C18H15NO3
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SMILES
O=C(C1=CC(OCC2=NC3=C(C=C2)C=CC=C3)=CC=C1)OC
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
CysLT1 receptor antagonist-1 Related Classifications
HY-165155 Related Classifications
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