AXL - AXL receptor tyrosine kinase Gene
Species: Bos taurus
Gene Type: protein coding
Gene ID: 516598
AXL Products (2)
| mRNA | Protein | Name |
|---|---|---|
| XM_024979095.1 | XP_024834863.1 | tyrosine-protein kinase receptor UFO isoform X1 |
| XM_024979096.1 | XP_024834864.1 | tyrosine-protein kinase receptor UFO isoform X2 |
| Protein Preferred Names | Protein Names | |
|---|---|---|
|
tyrosine-protein kinase receptor UFO |
|
Related Agents
- Approval
- Clinical Phase
- Pre-clinical Phase
Approval
Bioactive Molecules
(4)
| Cat. No. | Product Name |
Effect
|
Purity |
Rare Diseases
|
|---|---|---|---|---|
| HY-13016 | Cabozantinib | Inhibitor | 99.97% | Yes |
| HY-12432 | Gilteritinib | Inhibitor | 99.84% | Yes |
| HY-12432A | Gilteritinib hemifumarate | Inhibitor | 99.75% | Yes |
| HY-13016A | Cabozantinib hydrochloride | Inhibitor | / | Unkown |
Clinical Phase
Bioactive Molecules
(10)
| Cat. No. | Product Name |
Effect
|
Purity |
Phase |
|---|---|---|---|---|
| HY-138696 | Zanzalintinib | Inhibitor | 99.91% | Phase 3 |
| HY-15150 | Bemcentinib | Inhibitor | 99.92% | Phase 2 |
| HY-12076 | BMS 777607 | Inhibitor | 99.36% | Phase 2 |
| HY-12963 | Dubermatinib | Inhibitor | 99.84% | Phase 2 |
| HY-114358 | Tamnorzatinib | Inhibitor | 98.59% | Phase 2 |
| HY-107145A | Ningetinib | Inhibitor | 99.63% | Phase 2 |
| HY-107145 | Ningetinib Tosylate | Inhibitor | 99.59% | Phase 2 |
| HY-152830A | Adrixetinib TFA | Inhibitor | 99.82% | Phase 2 |
| HY-100946 | CEP-40783 | Inhibitor | 99.61% | Phase 1 |
| HY-147218 | PF-07265807 | Inhibitor | 95.18% | Phase 1 |
Bioactive MoleculesInhibitory Antibodies
(4)
| Cat. No. | Product Name |
Effect
|
Purity |
Phase |
|---|---|---|---|---|
| HY-P99463 | Batiraxcept | 99.91% | Phase 3 | |
| HY-P99360 | Enapotamab | Inhibitor | 99.9% | Phase 2 |
| HY-P99161 | Tilvestamab | Inhibitor | 98.08% | Phase 1 |
| HY-P991664 | AG01 | Inhibitor | 95.10% | Phase 1 |
Pre-clinical Phase
Bioactive Molecules
(46)
| Cat. No. | Product Name |
Effect
|
Purity |
Rare Diseases
|
|---|---|---|---|---|
| HY-114166 | 2-D08 | Inhibitor | 99.37% | Unkown |
| HY-15797 | UNC2250 | Inhibitor | 99.92% | Unkown |
| HY-12494 | LDC1267 | Inhibitor | 99.64% | Unkown |
| HY-117596 | UNC569 | Inhibitor | 99.92% | Unkown |
| HY-132200 | UNC5293 | Inhibitor | 99.93% | Unkown |
| HY-12964 | SGI-7079 | Inhibitor | 99.32% | Unkown |
| HY-100509 | NPS-1034 | Inhibitor | 98.0% | Unkown |
| HY-117548 | UNC1062 | Inhibitor | 98.92% | Unkown |
| HY-173268 | UNC9426 | Inhibitor | 99.51% | Unkown |
| HY-124066 | RU-302 | Inhibitor | 98.72% | Unkown |
| HY-15798 | UNC2881 | Inhibitor | 99.79% | Unkown |
| HY-124502 | UNC4203 | Inhibitor | 99.80% | Unkown |
| HY-152830 | Adrixetinib | Inhibitor | 99.55% | Unkown |
| HY-114357A | DS-1205b free base | Inhibitor | 99.92% | Unkown |
| HY-132893 | AZ14145845 | Inhibitor | 98.00% | Unkown |
| HY-144627 | PROTAC Axl Degrader 2 | Inhibitor | 98.01% | Unkown |
| HY-13016S | Cabozantinib-d6 | Inhibitor | 98.14% | Unkown |
| HY-151904 | AXL-IN-13 | Inhibitor | 98.03% | Unkown |
| HY-150041 | TL4830031 | Inhibitor | ≥98.0% | Unkown |
| HY-146615 | Axl-IN-6 | Inhibitor | / | Unkown |
| HY-152075 | AXL-IN-14 | Inhibitor | / | Unkown |
| HY-147574 | Axl-IN-7 | Inhibitor | / | Unkown |
| HY-147575 | Axl-IN-8 | Inhibitor | / | Unkown |
| HY-144708 | Axl-IN-4 | Inhibitor | / | Unkown |
| HY-144624 | PROTAC Axl Degrader 1 | Inhibitor | / | Unkown |
| HY-115778 | UNC3133 | Inhibitor | / | Unkown |
| HY-147578 | Axl-IN-11 | Inhibitor | / | Unkown |
| HY-176204 | Axl-IN-19 | Inhibitor | / | Unkown |
| HY-183774 | NTQ2494 | Inhibitor | / | Unkown |
| HY-153012 | Axl/Mer/CSF1R-IN-1 | Inhibitor | / | Unkown |
| HY-147576 | Axl-IN-9 | Inhibitor | / | Unkown |
| HY-15150G | Bemcentinib (GMP) | Inhibitor | / | Unkown |
| HY-184184 | Axl ligand-1 | Ligand | / | Unkown |
| HY-173400 | UNC8212 | Inhibitor | / | Unkown |
| HY-104075 | R916562 | Inhibitor | / | Unkown |
| HY-153441 | AXL-IN-15 | Inhibitor | / | Unkown |
| HY-147577 | Axl-IN-10 | Inhibitor | / | Unkown |
| HY-149092 | Anticancer agent 109 | / | Unkown | |
| HY-144706 | Axl-IN-3 | Inhibitor | / | Unkown |
| HY-147579 | Axl-IN-12 | Inhibitor | / | Unkown |
| HY-162085 | Axl-IN-17 | Inhibitor | / | Unkown |
| HY-122601 | TAM-IN-1 | Inhibitor | / | Unkown |
| HY-N12041 | Axl-IN-16 | Inhibitor | / | Unkown |
| HY-179535 | Axl-IN-21 | Inhibitor | / | Unkown |
| HY-146596 | Axl-IN-5 | Inhibitor | / | Unkown |
| HY-149491 | HIV-IN-7 | Inhibitor | / | Unkown |
Bioactive MoleculesInhibitory Antibodies
(3)
| Cat. No. | Product Name |
Effect
|
Purity |
Rare Diseases
|
|---|---|---|---|---|
| HY-P9988 | Mecbotamab | Inhibitor | 99.83% | Unkown |
| HY-P99733 | Mipasetamab | Inhibitor | 98.26% | Unkown |
| HY-P992116 | Ladarutatug | Inhibitor | 95.40% | Unkown |