L-803087 (Standard)
L-803087 (Standard) is the analytical standard of L-803087 (HY-108497). This product is intended for research and analytical applications. L-803087 is a potent and selective somatostatin sst4 receptor agonist with a Ki of 0.7 nM. L-803087 is >280-fold higher than other somatostatin receptors. L-803087 facilitates AMPA-mediated hippocampal synaptic responses in vitro and increases kainate-induced seizures in mice.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- CAS 番号: 217480-26-7
- 分子式: C25H29F2N5O3
- 分子量:485.53
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Product Information
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化学情報
- 純度とドキュメンテーション
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Help & FAQs
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HY-108497
L-803087sst4 Receptor Agonist -
HY-105172
TT-232SSTR1/SSTR4 Agonist -
HY-108498
L-817818Somatostatin Receptor Agonist -
HY-16381
PasireotideSomatostatin Agonist -
HY-108501
(1R,1'S,3'R/1R,1'R,3'S)-L-054,264sst2 Agonist -
HY-16381A
Pasireotide acetateSomatostatin Agonist -
HY-P1201
CyclosomatostatinSomatostatin Receptor Antagonist -
HY-P1206
CH 275SST1 Agonist -
HY-P1203
BIM-23056Somatostatin Receptor Antagonist -
HY-106103
Seglitidesomatostatin receptor Agonist Antagonist -
HY-108499
NNC 26-9100sst4 Agonist -
HY-P1212
Cortistatin 14 (mouse, rat)Neuropeptide
Product Information
説明
アプリケーション
The compound is the grade of analytical standard, which is the reference standard supplied assay. It is commonly used in qualitative, quantitative and methodological research experiments in HPLC, GC and MS.
化学情報
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CAS 番号 217480-26-7
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分子量 485.53
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分子式 C25H29F2N5O3
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SMILES
N=C(N)NCCC[C@@H](C(OC)=O)NC(CCCC1=C(C2=CC=CC=C2)NC3=C1C=C(F)C=C3F)=O
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
[1]. Rohrer SP, et al. Rapid identification of subtype-selective agonists of the somatostatin receptor through combinatorial chemistry. Science. 1998 Oct 23;282(5389):737-40. [Content Brief]
[2]. Moneta D, et al. Somatostatin receptor subtypes 2 and 4 affect seizure susceptibility and hippocampal excitatory neurotransmission in mice. Eur J Neurosci. 2002 Sep;16(5):843-9. [Content Brief]
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
L-803087 (Standard) 関連分類
HY-108497R 関連分類
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