2. Metabolic Enzyme/Protease
  3. Phosphodiesterase (PDE)
  4. Laprafylline

Laprafylline (S 9795), a xanthine derivative, is a bronchodilator. Laprafylline has potent anti-bronchoconstrictive effects, inhibiting action on mast cell degranulation and phosphodiesterase (PDE) activity (IC50 of 6 μM).

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Laprafylline

Laprafylline 화학구조

CAS No. : 90749-32-9

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제품 설명

Laprafylline (S 9795), a xanthine derivative, is a bronchodilator. Laprafylline has potent anti-bronchoconstrictive effects, inhibiting action on mast cell degranulation and phosphodiesterase (PDE) activity (IC50 of 6 μM)[1].

In Vivo

In male Sprague Dawley rats, Laprafylline (S 9795; 2.5-10mg/kg; iv) disappears rapidly from plasma with an elimination t1/2 of 0.8 h, regardless of the dose administered. The volume of distribution is high (about 3 L/kg) but total clearance is also high (about 40 mL/min/kg).

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
분자량

500.64

화학식

C29H36N6O2
CAS No.
SMILES

CC(C)CN1C2=C(C(N(C)C1=O)=O)N=C(CCN3CCN(C(C4=CC=CC=C4)C5=CC=CC=C5)CC3)N2
선적

Room temperature in continental US; may vary elsewhere.
보관

Please store the product under the recommended conditions in the Certificate of Analysis.
순도&문서
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Keywords:

Laprafylline90749-32-9S 9795S9795S-9795Phosphodiesterase (PDE)bronchodilatorxanthine derivativeanti-bronchoconstrictive effectsPDEInhibitorinhibitorinhibit

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Laprafylline
Cat. No.:
HY-106306
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