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Legumain inhibitor 1 

Cat. No.: HY-128617 Purity: 99.18% ee.: 100.00%
Handling Instructions

Legumain inhibitor 1 is a potent and selective Legumain inhibitor with an IC50 of 3.6 nM. Legumain inhibitor 1 can be used for cancer research.

For research use only. We do not sell to patients.

Legumain inhibitor 1 Chemical Structure

Legumain inhibitor 1 Chemical Structure

CAS No. : 2361157-34-6

Size Price Stock Quantity
Solution
10 mM * 1 mL in DMSO USD 514 In-stock
Estimated Time of Arrival: December 31
Solid + Solvent
10 mM * 1 mL
ready for reconstitution
USD 514 In-stock
Estimated Time of Arrival: December 31
Solid
5 mg USD 500 In-stock
Estimated Time of Arrival: December 31
10 mg USD 850 In-stock
Estimated Time of Arrival: December 31
25 mg USD 1800 In-stock
Estimated Time of Arrival: December 31
50 mg USD 3000 In-stock
Estimated Time of Arrival: December 31
100 mg USD 4600 In-stock
Estimated Time of Arrival: December 31
200 mg   Get quote  
500 mg   Get quote  

* Please select Quantity before adding items.

Customer Review

Based on 1 publication(s) in Google Scholar

Top Publications Citing Use of Products
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Description

Legumain inhibitor 1 is a potent and selective Legumain inhibitor with an IC50 of 3.6 nM. Legumain inhibitor 1 can be used for cancer research[1].

In Vitro

Legumain inhibitor 1 (Compound 16i) shows high microsomal stability with half-life’s in excess of 8 h (mouse and human MICs; CLint > 3 µL/min/mg)[1][1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

467.54

Formula

C₂₃H₂₅N₅O₄S

CAS No.
Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 40 mg/mL (85.55 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.1389 mL 10.6943 mL 21.3885 mL
5 mM 0.4278 mL 2.1389 mL 4.2777 mL
10 mM 0.2139 mL 1.0694 mL 2.1389 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: ≥ 5 mg/mL (10.69 mM); Clear solution

  • 2.

    Add each solvent one by one:  10% DMSO    90% (20% SBE-β-CD in saline)

    Solubility: ≥ 4 mg/mL (8.56 mM); Clear solution

  • 3.

    Add each solvent one by one:  10% DMSO    90% corn oil

    Solubility: ≥ 4 mg/mL (8.56 mM); Clear solution

*All of the co-solvents are provided by MCE.
References

Purity: 99.18% ee.: 100.00%

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This equation is commonly abbreviated as: C1V1 = C2V2

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Product Name:
Legumain inhibitor 1
Cat. No.:
HY-128617
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