MOR agonist-5
MOR agonist-5 is a selective and potent mu-opioid receptor (MOR) agonist with an EC50 of 0.25 nM. MOR agonist-5 shows an EC50 of 10 nM for DOR and >10000 nM for KOR and NOR. MOR agonist-5 exerts significant antinociceptive activity. MOR agonist-5 can be used for the research of pain.
For research use only. We do not sell to patients.
- CAS No.: 3085132-31-3
- Formula: C22H27N3O
- Molecular Weight:349.47
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All Opioid Receptor Isoforms
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Biological Activity
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μ Opioid Receptor/MOR 0.25 nM (EC50) |
δ Opioid Receptor/DOR 10 nM (EC50) |
κ Opioid Receptor/KOR >10000 nM (EC50) |
NOP Receptor/ORL1 >10000 nM (EC50) |
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 3085132-31-3
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Molecular Weight 349.47
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Formula C22H27N3O
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SMILES
NC(C1=CC(N2[C@H]3CC[C@@H]2CN(CCCC4=CC=CC=C4)C3)=CC=C1)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)