1. Membrane Transporter/Ion Channel
  2. Sodium Channel
  3. NaV1.7 inhibitor-1

NaV1.7 inhibitor-1 

Cat. No.: HY-119934
Handling Instructions

NaV1.7 inhibitor-1 is an efficacious voltage-gated sodium channel (NaV) 1.7 inhibitor with an IC50 of 0.6 nM for hNaV1.7, exhibits 80-fold selectivity versus hNaV1.5.

For research use only. We do not sell to patients.

NaV1.7 inhibitor-1 Chemical Structure

NaV1.7 inhibitor-1 Chemical Structure

CAS No. : 1494585-79-3

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Description

NaV1.7 inhibitor-1 is an efficacious voltage-gated sodium channel (NaV) 1.7 inhibitor with an IC50 of 0.6 nM for hNaV1.7, exhibits 80-fold selectivity versus hNaV1.5[1].

IC50 & Target

IC50: 0.6 nM (hNaV1.7)[1]

Molecular Weight

435.55

Formula

C₂₃H₃₀FNO₄S

CAS No.

1494585-79-3

SMILES

FC1=CC(OCC2(C)CCC3(CC3)CC2)=C(C4CC4)C=C1C(NS(C5CC5)(=O)=O)=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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NaV1.7 inhibitor-1
Cat. No.:
HY-119934
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